SCHEMBL10815751

SCHEMBL10815751

COc1ccc2c3c(c(=O)oc2c1OC)CN(CC(C)=O)CC3

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.70
DRD2 P14416 2/20 0.70
DRD3 P35462 1/20 0.70
MAOA P21397 6/20 0.58
MAOB P27338 6/20 0.58
ALDH1A1 P00352 7/20 0.53
HPGD P15428 5/20 0.53
MIF P14174 1/20 0.53
HDAC1 Q13547 1/20 0.52
KDM4E B2RXH2 5/20 0.52
HSD17B10 Q99714 4/20 0.52
TSHR P16473 3/20 0.52
ERN1 O75460 1/20 0.51
NPSR1 Q6W5P4 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
FHIT P49789 1/20 0.50
HTT P42858 2/20 0.43
LMNA P02545 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11759681 0.83 DRD4 (0.70) DRD4DRD2DRD3MAOAMAOB
SCHEMBL8583590 0.82 DRD4 (1.00) DRD4DRD2DRD3ALDH1A1HPGD
SCHEMBL11380048 0.81 DRD4 (0.66) DRD4DRD2DRD3MAOAMAOB
Hydrochloric Acid SCHEMBL10816670 0.80 DRD4 (0.65) DRD4DRD2DRD3MAOAMAOB
Hydrochloric Acid SCHEMBL10814338 0.80 DRD4 (0.65) DRD4DRD2DRD3MAOAMAOB
SCHEMBL10813145 0.79 DRD4 (0.66) DRD4DRD2DRD3ALDH1A1HPGD
SCHEMBL10813758 0.79 DRD4 (0.64) DRD4DRD2DRD3MAOAMAOB
SCHEMBL10813959 0.79 DRD4 (0.64) DRD4DRD2DRD3MAOAMAOB
SCHEMBL10817679 0.78 ERN1 (0.53) DRD4DRD2DRD3MAOAMAOB
SCHEMBL10815168 0.77 DRD4 (0.72) DRD4DRD2DRD3ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0087280-B1 3-(2-MONO-AND DIALKYLAMINO)PROPYL(-1,2,3,4-TETRAHYDRO-5H-(1) BENZOPYRANO(3,4-C)PYRIDIN-5-ONES AND DERIVATIVES THEREOF, A PROCESS FOR THEIR PRODUCTION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS WARNER-LAMBERT COMPANY (US) 1987-09-23 EP disclosed
EP-0087280-A2 3-(2-Mono-and dialkylamino)propyl(-1,2,3,4-tetrahydro-5H-(1) benzopyrano(3,4-c)pyridin-5-ones and derivatives thereof, a process for their production, and pharmaceutical compositions containing such compounds WARNER-LAMBERT COMPANY (US) 1983-08-31 EP disclosed
US-4382939-A 3-[2-(Mono-and dialkylamino)propyl]-1,2,3,4-tetrahydro-5H-[1]benzopyrano[3,4-C]pyridin-5-ones useful for treating bronchospastic diseases WARNER LAMBERT COMPANY (US) 1983-05-10 US disclosed