SCHEMBL10844762

SCHEMBL10844762

c1ccc(C(NCc2nccn2CC2CCNCC2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.39
GBA1 P04062 1/20 0.35
KDM1A O60341 6/20 0.34
MERTK Q12866 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 1/20 0.33
CYP2D6 P10635 1/20 0.33
HRH1 P35367 1/20 0.33
SCN1A P35498 1/20 0.33
SCN2A Q99250 1/20 0.33
SCN3A Q9NY46 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
MELK Q14680 1/20 0.32
AVPR2 P30518 1/20 0.32
AVPR1A P37288 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10845316 0.83 CHRM3 (0.34) MEN1KMT2A
SCHEMBL10846302 0.80 CHRM3 (0.34) MEN1KMT2A
SCHEMBL6152856 0.73 BRD4 (0.57) BRD4GBA1KDM1AMERTKMELK
SCHEMBL27798160 0.68 BRD4 (0.46) BRD4KDM1A
SCHEMBL1181466 0.67 BRD4 (0.55) BRD4KDM1AKMT2ACYP2D6
SCHEMBL27326515 0.66 BRD4 (0.46) BRD4KDM1A
Hydrochloric Acid SCHEMBL28784813 0.66 BRD4 (0.54) BRD4KDM1AKMT2ACYP2D6
SCHEMBL27490726 0.64 GBA1 (0.49) GBA1KDM1ACYP2D6MELK
Hydrochloric Acid SCHEMBL29957620 0.63 BRD4 (0.51) BRD4KDM1A
SCHEMBL10417634 0.63 BRD4 (0.43) BRD4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4605744-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1986-08-12 US disclosed
US-4537969-A AZOLE-SUBSTITUTED SATURATED HETEROCYCLIC CARBOXALDEHYDE ACETALS;INTERMEDIATES FOR 6-AMIDINOPENICILLINS HOFFMANN-LA ROCHE INC. (US) 1985-08-27 US disclosed
EP-0148283-A1 Novel penicillanic acid derivatives F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-07-17 EP disclosed
US-4431653-A ANTIBIOTICS; BACTERICIDES; SSYNERGISTIC WITH AMINO ACID DERIVATIVE HOFFMANN-LA ROCHE INC. (US) 1984-02-14 US disclosed