SCHEMBL10854343

SCHEMBL10854343

CCOC(=O)NC1CCc2ccccc2C1Nc1ccccc1CO

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.42
DRD2 P14416 1/20 0.38
TAS1R3 Q7RTX0 4/20 0.37
TAS1R1 Q7RTX1 4/20 0.37
TAS1R2 Q8TE23 4/20 0.37
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
KMT2A Q03164 3/20 0.35
HTT P42858 1/20 0.34
EPHX1 P07099 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10854332 1.00 ATM (0.42) ATMDRD2TAS1R3TAS1R1TAS1R2
SCHEMBL10854338 1.00 ATM (0.42) ATMDRD2TAS1R3TAS1R1TAS1R2
SCHEMBL10757437 0.89 ATM (0.51) ATMDRD2ALDH1A1HPGDSMN1; SMN2
SCHEMBL10757432 0.89 ATM (0.51) ATMDRD2ALDH1A1HPGDSMN1; SMN2
SCHEMBL7520297 0.89 ATM (0.42) ATMDRD2TAS1R3TAS1R1TAS1R2
SCHEMBL10921833 0.87 ATM (0.41) ATMTAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL10921832 0.87 ATM (0.41) ATMTAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL7370954 0.78 ATM (0.48) ATMALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL10759506 0.77 ATM (0.46) ATMALDH1A1HPGD
SCHEMBL10759500 0.77 ATM (0.46) ATMALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0088575-B1 PENTACYCLIC COMPOUNDS BEECHAM GROUP PLC (GB) 1986-12-30 EP disclosed
US-4585588-A ANTIDEPRESSANTS BEECHAM GROUP P.L.C. (GB) 1986-04-29 US disclosed
US-4504480-A DIAZABENZOCYCLOHEPTAFLUORENE DERIVATRIVES, ANTIDEPRESSANTS BEECHAM GROUP P.L.C. (GB) 1985-03-12 US disclosed