SCHEMBL10858748

SCHEMBL10858748

C=CC1(O)CCCc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.46
KDM1A O60341 3/20 0.44
AKR1B1 P15121 1/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TSHR P16473 2/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
DRD2 P14416 1/20 0.38
NFKB1 P19838 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR2B P41595 1/20 0.38
MTOR P42345 1/20 0.38
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10856627 0.89 KDM1A (0.42) SIGMAR1KDM1ATSHRHTR2AMAPK1
SCHEMBL11881410 0.78 ESR2 (0.41) KDM1ADRD2
SCHEMBL31629514 0.75 KDM1A (0.50) SIGMAR1KDM1AAKR1B1MEN1KMT2A
SCHEMBL4195493 0.75 KDM1A (0.50) SIGMAR1KDM1AAKR1B1MEN1KMT2A
SCHEMBL16388051 0.74 KDM1A (0.45) SIGMAR1KDM1ATSHRCYP3A4CYP2C19
SCHEMBL16924628 0.73 KDM1A (0.53) SIGMAR1KDM1ACYP3A4DRD2CYP2C19
SCHEMBL8659379 0.73 KDM1A (0.53) SIGMAR1KDM1ACYP3A4DRD2CYP2C19
SCHEMBL5533856 0.73 MAPK1 (0.42) SIGMAR1KDM1ACYP2D6HTR2AMAPK1
SCHEMBL11105463 0.72 KDM1A (0.42) SIGMAR1KDM1AAKR1B1MEN1KMT2A
SCHEMBL6689565 0.72 KDM1A (0.56) SIGMAR1KDM1AAKR1B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4590274-A Antihypertensive 1-[bis-(substituted phenyl)methyl]-4[2-(1,2,3,4-tetrahydro-substituted naphthalen-1-ylidene)ethyl]piperazines E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-05-20 US disclosed
EP-0069424-B1 PROCESS FOR THE SELECTIVE REDUCTION OF A 14, 17-DIOXO-8,4-SECO-STEROID AKZO N.V. (NL) 1985-05-29 EP disclosed
EP-0069424-A1 Process for the selective reduction of a 14, 17-dioxo-8,4-seco-steroid AKZO N.V. (NL) 1983-01-12 EP disclosed
US-4130565-A 3-ALKYL-TETRAHYDROPYRAN-OR THIOPYRAN-2,4-DIONES AS CHEMICAL INTERMEDIATES SHIONOGI & CO., LTD. (JP) 1978-12-19 US disclosed
US-4130565-A 3-ALKYL-TETRAHYDROPYRAN-OR THIOPYRAN-2,4-DIONES AS CHEMICAL INTERMEDIATES SHIONOGI & CO., LTD. (JP) 1978-12-19 US disclosed
US-4083852-A ORAL CONTRACEPTIVES SHIONOGI & CO., LTD. (JA) 1978-04-11 US disclosed