SCHEMBL10936216

SCHEMBL10936216

O=C(O)c1c[nH]c(Cc2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.50
GAA P10253 1/20 0.49
RAB9A P51151 1/20 0.49
NOTUM Q6P988 1/20 0.46
KDM5A P29375 2/20 0.44
KDM4C Q9H3R0 2/20 0.44
KDM5B Q9UGL1 2/20 0.44
KMT2A Q03164 2/20 0.43
KDM4A O75164 1/20 0.42
DAO P14920 2/20 0.42
PLA2G2A P14555 2/20 0.42
PLA2G10 O15496 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 2/20 0.41
SRD5A2 P31213 1/20 0.41
MEN1 O00255 1/20 0.41
HNF4A P41235 1/20 0.41
FOLH1 Q04609 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10941367 0.82 HPGD (0.42) HCAR2GAARAB9AKMT2ADAO
SCHEMBL7190682 0.81 ERCC5 (0.53) GAARAB9AKMT2ALMNAMEN1
SCHEMBL4671116 0.80 HCAR2 (0.39) HCAR2GAARAB9AKDM5AKDM4C
SCHEMBL4671120 0.80 HCAR2 (0.39) HCAR2GAARAB9AKDM5AKDM4C
SCHEMBL14604111 0.78 GAA (0.45) GAARAB9ANOTUMKMT2ADAO
SCHEMBL6613866 0.76 SMN1; SMN2 (0.57) HCAR2KDM5AKDM4CKDM5BKMT2A
SCHEMBL1584769 0.74 DAO (0.53) HCAR2KMT2ADAOMEN1
SCHEMBL25352675 0.73 NOTUM (0.52) HCAR2GAARAB9ANOTUMLMNA
SCHEMBL5158296 0.73 NOTUM (0.52) GAARAB9ANOTUMDAOLMNA
SCHEMBL27657375 0.73 NOTUM (0.52) GAARAB9ANOTUMDAOTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4511575-A Antidiabetic pyrrolecarboxylic acids PFIZER INC. (US) 1985-04-16 US disclosed
US-4511576-A Antidiabetic pyrrolecarboxylic acids PFIZER INC. (US) 1985-04-16 US disclosed
US-4351843-A LOWERING BLOOD GLUCOSE PFIZER INC. (US) 1982-09-28 US disclosed
US-4282242-A HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1981-08-04 US disclosed