SCHEMBL10965014

SCHEMBL10965014

[c]1ccncc1-c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 12/20 0.56
CYP3A4 P08684 4/20 0.56
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 1/20 0.56
KDM4E B2RXH2 2/20 0.48
HPGD P15428 2/20 0.48
HSD17B10 Q99714 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CYP2B6 P20813 4/20 0.46
CYP2C9 P11712 3/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2E1 P05181 3/20 0.42
MKNK1 Q9BUB5 2/20 0.41
MKNK2 Q9HBH9 2/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL386070 0.85 CYP2A6 (0.41) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL38500 0.82 CYP2A6 (0.54) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL7875042 0.78 MAPT (0.43) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL6104498 0.76 CYP2A6 (0.47) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL10852859 0.76 CYP2A6 (0.47) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL11358625 0.76 CYP2A6 (0.51) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL9958676 0.76 CYP19A1 (0.50) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL5544009 0.76 IDO1 (0.44) CYP3A4KDM4ETP53CYP11B2
SCHEMBL29419014 0.74 CYP2A6 (1.00) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL30473120 0.74 CYP2A6 (1.00) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154190-A1 Pyridones MERCK PATENT GmbH (DE) 1985-09-11 EP disclosed