SCHEMBL10976554

SCHEMBL10976554

Oc1ccc(Nc2ncc(-c3ccc(O)cc3)cn2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
KMT2A Q03164 1/20 0.55
AURKA O14965 11/20 0.53
SYK P43405 1/20 0.53
CSNK2A1 P68400 1/20 0.51
CHEK1 O14757 1/20 0.45
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
VCP P55072 2/20 0.44
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
AMY1A P0DUB6 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
THRB P10828 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10979289 0.91 GFRA3 (0.51) MEN1NPC1RAB9AKMT2AAURKA
SCHEMBL5496551 0.81 CTSC (0.44) AURKASYK
SCHEMBL12846706 0.81 CSNK2A1 (0.50) MEN1NPC1RAB9AKMT2AAURKA
SCHEMBL11455773 0.80 MAPT (0.56) MEN1NPC1RAB9AKMT2AAURKA
SCHEMBL12179363 0.79 ESR2 (0.50) MEN1NPC1RAB9AKMT2AAURKA
SCHEMBL1921278 0.78 ESR1 (0.65) MEN1NPC1RAB9AKMT2AESR1
SCHEMBL13605301 0.77 RIPK2 (0.61) ESR1ESR2
SCHEMBL4498501 0.77 AURKA (0.63) MEN1NPC1RAB9AKMT2AAURKA
SCHEMBL5501103 0.77 MAPT (0.52) MEN1NPC1KMT2AAURKASYK
SCHEMBL10971409 0.76 HDAC3 (0.59) MEN1NPC1RAB9AKMT2AAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0164204-A1 Novel pharmaceutically useful pyrimidines FISONS plc (GB) 1985-12-11 EP claimed
EP-0164204-A1 Novel pharmaceutically useful pyrimidines FISONS plc (GB) 1985-12-11 EP disclosed