SCHEMBL10994860

SCHEMBL10994860

Cc1[nH]c(=O)c(N)cc1-c1ccc(N)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 4/20 0.75
PDE3A Q14432 4/20 0.75
PDE4A P27815 2/20 0.75
PDE4B Q07343 2/20 0.75
PDE4C Q08493 2/20 0.75
PDE4D Q08499 2/20 0.75
AURKB Q96GD4 1/20 0.71
INCENP Q9NQS7 1/20 0.71
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
GALR3 O60755 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
PDE5A O76074 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
PTGS1 P23219 1/20 0.42
CYP2C19 P33261 1/20 0.42
BLM P54132 1/20 0.42
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10989420 0.86 PDE3B (0.71) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL8207560 0.86 PDE3B (1.00) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10997163 0.83 PDE3B (0.67) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11235286 0.83 PDE3B (1.00) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10995497 0.81 PDE3B (0.63) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10992753 0.80 PDE3B (0.62) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11002239 0.79 PDE3B (0.49) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10891425 0.79 KDM4E (0.73) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10478089 0.79 PDE3B (0.85) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10998080 0.78 PDE3B (0.59) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4559352-A 1,2-Dihydro-2-oxo-5-(hydroxy-and/or amino-phenyl)-nicotinonitriles and cardiotonic use thereof STERLING DRUG INC. (US) 1985-12-17 US disclosed
US-4515797-A 3-Amino-5-(hydroxy- and/or aminophenyl)-6-(lower-alkyl)-2(1H)-pyridinones and cardiotonic use thereof STERLING DRUG INC. (US) 1985-05-07 US disclosed
EP-0061774-A2 3-Amino-5-(substituted)-2 (1H) pyridinones and 3-cyano compounds useful as cardiotonics and preparation thereof STERLING DRUG INC. (US) 1982-10-06 EP disclosed