SCHEMBL10997396

SCHEMBL10997396

CCOC(=O)c1cnc2sc(C)cc2c1Cl

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
HPGD P15428 5/20 0.44
MAPT P10636 4/20 0.44
RECQL P46063 2/20 0.44
NPSR1 Q6W5P4 1/20 0.43
DPP4 P27487 2/20 0.42
BAZ2B Q9UIF8 1/20 0.42
BAZ2A Q9UIF9 1/20 0.42
ALDH1A1 P00352 5/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 2/20 0.41
PKM P14618 1/20 0.41
MAPK10 P53779 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22917929 0.86 KMT2A (0.50) KMT2AMEN1HPGDMAPTRECQL
SCHEMBL10998213 0.86 MAPT (0.46) HPGDMAPTRECQLDPP4ALDH1A1
SCHEMBL10812459 0.80 CUL4A (0.42) KMT2AMEN1HPGDMAPTRECQL
SCHEMBL4906865 0.80 KMT2A (0.54) KMT2AMEN1HPGDMAPTRECQL
SCHEMBL12533457 0.78 CDC7 (0.43) KMT2AMEN1HPGDMAPTNPSR1
SCHEMBL11578876 0.78 MAPT (0.49) KMT2AMEN1HPGDMAPTRECQL
SCHEMBL5929779 0.77 KMT2A (0.54) KMT2AMEN1HPGDMAPTNPSR1
SCHEMBL31513547 0.77 KMT2A (0.51) KMT2AMEN1HPGDMAPTRECQL
SCHEMBL19814475 0.77 KMT2A (0.51) KMT2AMEN1HPGDMAPTRECQL
SCHEMBL25656120 0.76 KMT2A (0.53) KMT2AMEN1MAPTNPSR1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100168123-A1 AKT PROTEIN KINASE INHIBITORS ARRAY BIOPHARMA INC. 2010-07-01 US disclosed
US-4560689-A ANTICONVULSANTS, ANTIDEPRESSANTS, SEDATIVE ANTIDOTES, AND ANTIEPLILEPTIC AGENTS CIBA-GEIGY CORPORATION (US) 1985-12-24 US disclosed
US-4479955-A ANTICONVULSANTS, ANTIDEPRESSANTS, ANTIEPILEPTIC AGENTS CIBA-GEIGY CORPORATION (US) 1984-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168123-A1 AKT PROTEIN KINASE INHIBITORS AKT1, AKT2, AKT3 KMT2A 2166/4885MEN1 2997/4885HPGD 3893/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.