SCHEMBL10999940

SCHEMBL10999940

Cc1ccc(C2CN(C)Cc3sc(Br)cc32)cc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.57
SLC6A2 P23975 17/20 0.57
SLC6A3 Q01959 17/20 0.57
CYP2D6 P10635 1/20 0.49
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
DRD1 P21728 1/20 0.41
HRH3 Q9Y5N1 1/20 0.39
KIF11 P52732 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11218070 0.90 NPC1 (0.47) SLC6A4SLC6A2SLC6A3CYP2D6NPC1
SCHEMBL11214213 0.87 SLC6A2 (0.55) SLC6A4SLC6A2SLC6A3CYP2D6DRD1
SCHEMBL11215925 0.84 SLC6A2 (0.56) SLC6A4SLC6A2SLC6A3CYP2D6NPC1
SCHEMBL10999076 0.82 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3CYP2D6NPC1
SCHEMBL11000109 0.82 SLC6A2 (0.46) SLC6A4SLC6A2SLC6A3CYP2D6NPC1
Bromide SCHEMBL11038410 0.81 NPC1 (0.68) SLC6A4SLC6A2SLC6A3NPC1RAB9A
SCHEMBL11003203 0.81 SLC6A4 (0.52) SLC6A4SLC6A2SLC6A3CYP2D6NPC1
Hydrochloric Acid SCHEMBL11222430 0.81 SLC6A2 (0.45) SLC6A4SLC6A2SLC6A3CYP2D6NPC1
SCHEMBL11004967 0.79 NPC1 (0.45) SLC6A4SLC6A2SLC6A3CYP2D6NPC1
SCHEMBL11215415 0.78 SLC6A2 (0.44) SLC6A4SLC6A2SLC6A3CYP2D6NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4550106-A ANTIDEPRESSANTS BOEHRINGER INGELHEIM KG (DE) 1985-10-29 US disclosed
US-4482559-A ANTIDEPRESSANT BOEHRINGER INGELHEIM KG (DE) 1984-11-13 US disclosed
US-4322423-A 4-Phenyl-4,5,6,7-tetrahydro-thieno(2,3-C)pyridines and salts thereof BOEHRINGER INGELHEIM GMBH (DE) 1982-03-30 US disclosed