SCHEMBL11001240

SCHEMBL11001240

COc1ccc([C@H]2Sc3ccccc3N(CCN(C)C)C(=O)[C@H]2OC(=O)c2ccccc2[N+](=O)[O-])cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1S Q13698 10/20 0.72
CYP3A4 P08684 3/20 0.72
TSHR P16473 2/20 0.72
ABCB11 O95342 2/20 0.72
LMNA P02545 2/20 0.72
KCNH2 Q12809 2/20 0.72
CACNA1C Q13936 2/20 0.72
SLC22A1 O15245 1/20 0.72
CACNA1F O60840 1/20 0.72
ABCB1 P08183 1/20 0.72
HRH2 P25021 1/20 0.72
ADRA1A P35348 1/20 0.72
SCN1A P35498 1/20 0.72
SCN4A P35499 1/20 0.72
HTT P42858 1/20 0.72
SCN7A Q01118 1/20 0.72
CACNA1D Q01668 1/20 0.72
PLAUR Q03405 1/20 0.72
SCN5A Q14524 1/20 0.72
SCN9A Q15858 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11117127 1.00 CACNA1S (0.72) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL11006691 0.92 CACNA1S (0.67) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL11006682 0.92 CACNA1S (0.67) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL11006686 0.92 CACNA1S (0.67) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10504834 0.91 CACNA1S (0.66) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL11003409 0.91 CACNA1S (0.66) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10504950 0.91 CACNA1S (0.66) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10504944 0.91 CACNA1S (0.66) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10504829 0.91 CACNA1S (0.66) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10504824 0.91 CACNA1S (0.66) CACNA1SCYP3A4TSHRABCB11LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521430-A VASODILATOR, ANTIISCHEMIC AGENT TANABE SEIYAKU CO., LTD. (JP) 1985-06-04 US disclosed
EP-0128462-A1 Novel benzothiazepine derivatives, processes for preparing the same and pharmaceutical compositions Tanabe Seiyaku Co., Ltd. (JP) 1984-12-19 EP disclosed