SCHEMBL11004166

SCHEMBL11004166

COC(=O)C(=Cc1ccccc1OC(F)(F)F)C(C)=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MEN1 O00255 1/20 0.45
PLIN1 O60240 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
PLIN5 Q00G26 1/20 0.45
KMT2A Q03164 1/20 0.45
ABHD5 Q8WTS1 1/20 0.45
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GAA P10253 1/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
CYP1A2 P05177 1/20 0.40
HIF1A Q16665 1/20 0.40
ANO1 Q5XXA6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11004161 1.00 MAPT (0.46) MAPTNPSR1MEN1PLIN1LMNA
SCHEMBL10353470 0.84 MAPT (0.61) MAPTNPSR1MEN1PLIN1LMNA
SCHEMBL11002399 0.84 MAPT (0.61) MAPTNPSR1MEN1PLIN1LMNA
SCHEMBL9386421 0.80 MAPT (0.48) MAPTNPSR1MEN1LMNAKMT2A
SCHEMBL10744797 0.80 MAPT (0.48) MAPTNPSR1MEN1LMNAKMT2A
SCHEMBL10481034 0.80 MAPT (0.48) MAPTNPSR1MEN1LMNAKMT2A
SCHEMBL7378695 0.78 CYP1A2 (0.63) MAPTNPSR1MEN1PLIN1LMNA
SCHEMBL7378697 0.78 CYP1A2 (0.63) MAPTNPSR1MEN1PLIN1LMNA
SCHEMBL1508463 0.77 AKR1C3 (0.47) LMNAPOLBKMT2AALDH1A1L3MBTL1
SCHEMBL1508462 0.77 AKR1C3 (0.47) LMNAPOLBKMT2AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4532248-A Administering 1,4-dihydropyridine derivative exhibiting positive inotropic activity BAYER AKTIENGESELLSCHAFT (DE) 1985-07-30 US disclosed