SCHEMBL11005523

SCHEMBL11005523

COc1ccc(C2CN(C)Cc3sc(CO)cc32)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SLC6A4 P31645 7/20 0.39
SLC6A2 P23975 6/20 0.39
SLC6A3 Q01959 6/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11005340 0.86 SLC6A4 (0.47) SLC6A4SLC6A2SLC6A3HRH3
SCHEMBL11037531 0.82 NPC1 (0.43) NPC1RAB9ASLC6A4SLC6A2SLC6A3
SCHEMBL11006639 0.82 NPC1 (0.65) NPC1RAB9ASLC6A4SLC6A2SLC6A3
SCHEMBL11003203 0.82 SLC6A4 (0.52) NPC1RAB9ASLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL11035959 0.81 NPC1 (0.43) NPC1RAB9ASLC6A4SLC6A2SLC6A3
SCHEMBL11005771 0.81 SLC6A4 (0.50) NPC1RAB9ASLC6A4SLC6A2SLC6A3
SCHEMBL11003392 0.81 SLC6A4 (0.50) NPC1RAB9ASLC6A4SLC6A2SLC6A3
SCHEMBL11038643 0.79 NPC1 (0.64) NPC1RAB9ASLC6A4SLC6A2SLC6A3
SCHEMBL11000917 0.73 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3HRH3
SCHEMBL11000635 0.72 SLC6A4 (0.48) NPC1RAB9ASLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4550106-A ANTIDEPRESSANTS BOEHRINGER INGELHEIM KG (DE) 1985-10-29 US disclosed
US-4482559-A ANTIDEPRESSANT BOEHRINGER INGELHEIM KG (DE) 1984-11-13 US disclosed
EP-0088250-A2 Basic substituted 4-phenyl-4,5,6,7-tetrahydrothieno(2,3-c) pyridines, process for their preparation and pharmaceutical compositions containing them BOEHRINGER INGELHEIM KG (DE) 1983-09-14 EP disclosed