SCHEMBL11012000

SCHEMBL11012000

C=C(CC)Sc1ccc(-c2nc3ncncc3[nH]2)c(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.42
ENPP1 P22413 1/20 0.40
PDE5A O76074 11/20 0.39
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AURKA O14965 1/20 0.38
NPY5R Q15761 1/20 0.37
METAP2 P50579 1/20 0.37
METAP1 P53582 1/20 0.37
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11233387 0.83 PDE2A (0.48) PDE2AENPP1PDE5APDE3BPDE3A
SCHEMBL11009401 0.81 ENPP1 (0.43) PDE2AENPP1PDE5APDE3BPDE3A
SCHEMBL11009066 0.81 ENPP1 (0.52) PDE2AENPP1PDE5APDE3BPDE3A
SCHEMBL11012152 0.80 ENPP1 (0.53) PDE2AENPP1PDE5APDE3BPDE3A
SCHEMBL11008089 0.79 ENPP1 (0.48) PDE2AENPP1PDE5APDE3BPDE3A
SCHEMBL11010105 0.79 ENPP1 (0.43) PDE2AENPP1PDE5APDE3BPDE3A
SCHEMBL10749457 0.78 PDE2A (0.50) PDE2AENPP1PDE5APDE3BPDE3A
Hydrochloric Acid SCHEMBL11272588 0.78 PDE5A (0.45) PDE2AENPP1PDE5APDE3BPDE3A
SCHEMBL11006136 0.78 PDE2A (0.42) PDE2AENPP1PDE5APDE3BPDE3A
Hydrochloric Acid SCHEMBL11238238 0.77 PDE2A (0.49) PDE2AENPP1PDE5APDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142075-A2 Purine derivatives, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-05-22 EP disclosed