SCHEMBL11015992

SCHEMBL11015992

COC(=O)c1ccc2c(c1)Sc1cc(N)ccc1C=C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.46
KDM4E B2RXH2 6/20 0.46
HSD17B10 Q99714 5/20 0.46
ALDH1A1 P00352 5/20 0.46
HPGD P15428 4/20 0.46
GAA P10253 3/20 0.46
CASP1 P29466 2/20 0.46
CASP7 P55210 2/20 0.46
GLA P06280 1/20 0.46
ATM Q13315 1/20 0.46
MAPK1 P28482 3/20 0.46
PTPRC P08575 1/20 0.44
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
XDH P47989 1/20 0.42
NOX1 Q9Y5S8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10979797 0.82 MAPT (0.46) MAPTKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL10978657 0.81 NOX1 (0.46) MAPTKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL69897 0.76 CA1 (0.55) MAPTKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9508150 0.76 CA1 (0.55) MAPTKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL11100052 0.75 NOX1 (0.40) MAPTKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL2880869 0.75 PTPRC (0.49) MAPTKDM4EHSD17B10ALDH1A1HPGD
Hydrochloric Acid SCHEMBL5193420 0.73 PTPRC (0.48) MAPTKDM4EHSD17B10ALDH1A1HPGD
Hydrochloric Acid SCHEMBL11015056 0.73 NOX1 (0.39) MAPTKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9295482 0.73 PTPRC (0.62) MAPTKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL2330668 0.73 PLAU (0.61) MAPTKDM4EHSD17B10ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4536507-A ANTIASTHMA AGENTS MERCK & CO., INC. (US) 1985-08-20 US disclosed
EP-0052912-A1 7-Fluoro-dibenzo(b,f)thiepin derivatives, their preparation and resolution, and compositions containing them MERCK & CO. INC. (US) 1982-06-02 EP disclosed