SCHEMBL1101657

SCHEMBL1101657

CCOC(=O)c1cc(C)c(N)c(C)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.60
CA1 P00915 3/20 0.60
CA2 P00918 3/20 0.60
CA7 P43166 3/20 0.60
CA9 Q16790 3/20 0.60
CA14 Q9ULX7 3/20 0.60
CYP3A4 P08684 2/20 0.58
LMNA P02545 1/20 0.58
CYP1A2 P05177 1/20 0.58
MAOA P21397 1/20 0.58
NPC1 O15118 2/20 0.53
ESR1 P03372 3/20 0.50
ESR2 Q92731 1/20 0.50
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 4/20 0.46
GAA P10253 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
MAPT P10636 3/20 0.46
KDM4E B2RXH2 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8284687 0.91 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL17955668 0.89 CA12 (0.53) CA12CA1CA2CA7CA9
SCHEMBL28572600 0.88 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL10146774 0.88 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL1664013 0.83 CA12 (0.75) CA12CA1CA2CA7CA9
SCHEMBL7929919 0.82 CA1 (0.58) CA12CA1CA2CA7CA9
SCHEMBL1278720 0.82 NPC1 (0.68) CA12CA1CA2CA7CA9
SCHEMBL869061 0.82 ESR1 (0.71) CA12CA1CA2CA7CA9
SCHEMBL28692452 0.82 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL2810136 0.82 NPC1 (0.68) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 67 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023114977-A1 S1PR4 RECEPTOR ANTAGONISTS AND METHODS OF USE THEREOF TIAKI THERAPEUTICS, INC. (US) 2023-06-22 WO disclosed
EP-3808743-A1 HIV REPLICATION INHIBITING PYRIMIDINES Janssen Pharmaceutica NV (BE) 2021-04-21 EP disclosed
CN-108034395-B LED lens fixing UV glue and preparation method and application thereof 广州惠利电子材料有限公司 2020-11-10 CN disclosed
EP-3083554-B1 DIMETHYLBENZOIC ACID COMPOUNDS LILLY CO ELI (US) 2019-03-13 EP disclosed
US-10077270-B2 HIV inhibiting bicyclic pyrimidine derivatives JANSSEN SCIENCES IRELAND UC (IE) 2018-09-18 US disclosed
US-10072015-B2 HIV inhibiting bicyclic pyrimidine derivatives JANSSEN SCIENCES IRELAND UC (IE) 2018-09-11 US disclosed
US-10005721-B2 Dimethylbenzoic acid compounds ELI LILLY AND COMPANY (US) 2018-06-26 US disclosed
US-9926276-B2 Substituted benzamides with activity towards EP4 receptors DRACONIS PHARMA, S.L. (ES) 2018-03-27 US disclosed
US-20180016281-A1 HIV INHIBITING BICYCLIC PYRIMIDINE DERIVATIVES JANSSEN SCIENCES IRELAND UC (IE) 2018-01-18 US disclosed
US-20180016281-A1 HIV INHIBITING BICYCLIC PYRIMIDINE DERIVATIVES JANSSEN SCIENCES IRELAND UC (IE) 2018-01-18 US disclosed
EP-0661350-B1 Quinizarin compound, method for production thereof, and use therefor NIPPON CATALYTIC CHEM IND (JP) 2001-08-22 EP disclosed
EP-0632038-B1 METHOTREXATE DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 2001-08-22 EP disclosed
US-5968688-A RESINS AND DYES FOR COLOR FILTERS NIPPON SHOKUBAI CO., LTD. (JP) 1999-10-19 US disclosed
US-5817843-A Quinizarin compound, method for production thereof, and use therefor NIPPON SHOKUBAI CO., LTD. (JP) 1998-10-06 US disclosed
CN-1039907-C Methotrexate derivative CHUGAI PHARMACEUTICAL CO LTD (JP) 1998-09-23 CN disclosed
EP-0833203-A1 Color filter grade photosensitive resin coloring composition, and color filter using the same NIPPON SHOKUBAI CO., LTD. (JP) 1998-04-01 EP disclosed
US-5608091-A SHEETS FOR HEAT EXCHANGING AND OPTICAL RECORDING MATERIAL NIPPON SHOKUBAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0661350-A1 Quinizarin compound, method for production thereof, and use therefor NIPPON SHOKUBAI CO., LTD. (JP) 1995-07-05 EP disclosed
EP-0632038-A1 METHOTREXATE DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 1995-01-04 EP disclosed
CN-1077956-A METHOTREXATE DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 1993-11-03 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10072015-B2 HIV inhibiting bicyclic pyrimidine derivatives ZC3HAV1, CCR6, ZC3HAV1L CA12 4782/4885CA1 4496/4885CA2 4509/4885
US-20180016281-A1 HIV INHIBITING BICYCLIC PYRIMIDINE DERIVATIVES COX6C, ZC3HAV1L, CCR6 CA12 4775/4885CA1 4538/4885CA2 4369/4885
US-10077270-B2 HIV inhibiting bicyclic pyrimidine derivatives ZC3HAV1, CCR6, COX6C CA12 4766/4885CA1 4501/4885CA2 4549/4885
US-10005721-B2 Dimethylbenzoic acid compounds PTGER4, EDNRB, EPB41 CA12 2690/4885CA1 2400/4885CA2 567/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.