SCHEMBL11022069

SCHEMBL11022069

CN(C)C1=NC(c2ccc(Br)cc2)c2ccccc2C1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.43
HTR2A P28223 10/20 0.43
HTR2C P28335 7/20 0.43
HTR2B P41595 6/20 0.43
HRH3 Q9Y5N1 6/20 0.43
KCNH2 Q12809 1/20 0.36
HRH1 P35367 3/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10857223 0.97 HTR2A (0.44) SMN1; SMN2HTR2AHTR2CHTR2BHRH3
SCHEMBL11018524 0.86 HTR2A (0.44) HTR2AHTR2CHTR2BHRH3KCNH2
Hydrochloric Acid SCHEMBL10857042 0.85 KCNH2 (0.44) HTR2AHTR2CHTR2BHRH3KCNH2
Hydrochloric Acid SCHEMBL10857036 0.85 KCNH2 (0.44) HTR2AHTR2CHTR2BHRH3KCNH2
Hydrochloric Acid SCHEMBL10850138 0.83 HTR2A (0.44) HTR2AHTR2CHTR2BHRH3KCNH2
SCHEMBL11016226 0.82 HTR2A (0.40) HTR2AHTR2CHTR2BHRH3HRH1
SCHEMBL11018044 0.82 KCNH2 (0.34) HTR2AKCNH2HRH1SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL10855338 0.81 SRD5A2 (0.38) HTR2AKCNH2HRH1MEN1NPC1
Hydrochloric Acid SCHEMBL10855971 0.81 KCNH2 (0.34) HTR2AKCNH2HRH1SLC6A4NPC1
Hydrochloric Acid SCHEMBL10856997 0.81 KCNH2 (0.34) HTR2AKCNH2HRH1SLC6A4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0139296-A2 Dihydroisoquinoline derivatives BEECHAM GROUP PLC (GB) 1985-05-02 EP claimed