SCHEMBL11043930

SCHEMBL11043930

c1ccc2c(c1)C[C@H]1CCc3ccccc3[C@H]1O2

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.41
CHRM4 P08173 2/20 0.41
CHRM5 P08912 2/20 0.41
CHRM1 P11229 2/20 0.41
CHRM3 P20309 2/20 0.41
SIGMAR1 Q99720 3/20 0.40
IDO1 P14902 2/20 0.40
PDPK1 O15530 1/20 0.40
CYP11B2 P19099 1/20 0.38
CHRNA7 P36544 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11043928 1.00 CHRM2 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11042908 1.00 CHRM2 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11043767 0.85 CHRM2 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11046975 0.85 CHRM2 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11049212 0.84 CYP19A1 (0.38) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11049210 0.84 CYP19A1 (0.38) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11352506 0.84 CYP19A1 (0.38) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11045163 0.84 HRH4 (0.41) CHRM2SIGMAR1
SCHEMBL11364253 0.84 HRH4 (0.41) CHRM2SIGMAR1
SCHEMBL11045161 0.84 HRH4 (0.41) CHRM2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0025599-B1 BENZOPYRAN COMPOUNDS, USEFUL AS CHEMOTHERAPEUTIC AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1984-12-19 EP disclosed
US-4452991-A OR BENZO(B)INDENO (2,1-E) PYRANS OR BENZO(C)XANTHENES BATCHELOR JOHN F (GB) 1984-06-05 US disclosed
EP-0025599-A1 Benzopyran compounds, useful as chemotherapeutic agents THE WELLCOME FOUNDATION LIMITED (GB) 1981-03-25 EP disclosed