SCHEMBL11044525

SCHEMBL11044525

Clc1ccc2c(c1)C[C@H]1Cc3ccccc3O[C@@H]21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.45
CYP19A1 P11511 4/20 0.41
TRPM5 Q9NZQ8 2/20 0.39
TRPM4 Q8TD43 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
MAOB P27338 1/20 0.38
CHRM2 P08172 3/20 0.38
CHRM4 P08173 2/20 0.38
CHRM5 P08912 2/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 2/20 0.38
AR P10275 1/20 0.37
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11042094 0.90 HTR2C (0.47) HTR2CCYP19A1TRPM5TRPM4HRH4
SCHEMBL11049212 0.88 CYP19A1 (0.38) HTR2CCYP19A1HRH4HRH3MAOB
SCHEMBL11352506 0.88 CYP19A1 (0.38) HTR2CCYP19A1HRH4HRH3MAOB
SCHEMBL11049210 0.88 CYP19A1 (0.38) HTR2CCYP19A1HRH4HRH3MAOB
SCHEMBL11046135 0.88 HRH3 (0.45) HTR2CCYP19A1TRPM5HRH4HRH3
SCHEMBL11043767 0.81 CHRM2 (0.41) HRH3MAOBCHRM2CHRM4CHRM5
SCHEMBL11046975 0.81 CHRM2 (0.41) HRH3MAOBCHRM2CHRM4CHRM5
SCHEMBL11045163 0.80 HRH4 (0.41) HTR2CHRH4HRH3MAOBCHRM2
SCHEMBL11364253 0.80 HRH4 (0.41) HTR2CHRH4HRH3MAOBCHRM2
SCHEMBL11045161 0.80 HRH4 (0.41) HTR2CHRH4HRH3MAOBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452991-A OR BENZO(B)INDENO (2,1-E) PYRANS OR BENZO(C)XANTHENES BATCHELOR JOHN F (GB) 1984-06-05 US claimed
EP-0025599-B1 BENZOPYRAN COMPOUNDS, USEFUL AS CHEMOTHERAPEUTIC AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1984-12-19 EP disclosed
US-4452991-A OR BENZO(B)INDENO (2,1-E) PYRANS OR BENZO(C)XANTHENES BATCHELOR JOHN F (GB) 1984-06-05 US disclosed
EP-0025599-A1 Benzopyran compounds, useful as chemotherapeutic agents THE WELLCOME FOUNDATION LIMITED (GB) 1981-03-25 EP disclosed