SCHEMBL11048112

SCHEMBL11048112

COc1ccc(Cl)cc1C1(O)C(=O)NC(=O)NC1=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 3/20 0.47
MMP3 P08254 1/20 0.47
MMP8 P22894 1/20 0.47
MMP14 P50281 1/20 0.47
MMP17 Q9ULZ9 1/20 0.47
KCNQ3 O43525 1/20 0.46
KCNQ2 O43526 1/20 0.46
KCNQ4 P56696 1/20 0.46
KCNMA1 Q12791 1/20 0.46
KCNQ5 Q9NR82 1/20 0.46
KMT2A Q03164 2/20 0.46
ADAM17 P78536 2/20 0.43
ADAMTS5 Q9UNA0 2/20 0.43
MMP13 P45452 2/20 0.43
AKR1B1 P15121 4/20 0.42
AKR1A1 P14550 1/20 0.42
IDO1 P14902 1/20 0.40
MEN1 O00255 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2495393 0.85 KMT2A (0.57) MMP2MMP3MMP8MMP14MMP17
SCHEMBL11042537 0.83 KMT2A (0.47) MMP2MMP3MMP8MMP14MMP17
SCHEMBL11070824 0.82 KMT2A (0.49) KMT2AAKR1B1AKR1A1HTR2AHTR2C
SCHEMBL2497429 0.80 CBX7 (0.52) KCNQ3KCNQ2KCNQ4KCNMA1KCNQ5
SCHEMBL2497604 0.80 KMT2A (0.51) MMP2MMP3MMP8MMP14MMP17
SCHEMBL5982243 0.80 KCNQ3 (0.46) MMP2MMP3MMP8MMP14MMP17
SCHEMBL2499035 0.79 KMT2A (0.53) KCNQ3KCNQ2KCNQ4KCNMA1KCNQ5
SCHEMBL5860255 0.79 KMT2A (0.50) KCNQ3KCNQ2KCNQ4KCNMA1KCNQ5
SCHEMBL5857998 0.79 KMT2A (0.53) MMP2MMP3MMP8MMP14MMP17
SCHEMBL5858048 0.79 KMT2A (0.50) MMP2MMP3MMP8MMP14MMP17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4454320-A Process for 5-substituted dialuric acids PFIZER INC. (US) 1984-06-12 US disclosed
US-4448971-A Hypoglycemic 5-phenyl-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1984-05-15 US disclosed
US-4407811-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1983-10-04 US disclosed
US-4367234-A HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1983-01-04 US disclosed