SCHEMBL11054308

SCHEMBL11054308

CNC(=O)N(C(=N)N)c1c(C)cc(N)cc1Cl

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.32
THRB P10828 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11061869 0.90 KDM4E (0.33)
Hydrochloric Acid SCHEMBL11505528 0.88 KDM4E (0.32)
SCHEMBL11058712 0.87 CYP3A4 (0.35) CYP3A4
SCHEMBL11058085 0.85 CA1 (0.31) CA1CA2
SCHEMBL11225624 0.84 POLB (0.32)
Hydrochloric Acid SCHEMBL11134530 0.83 POLB (0.31)
SCHEMBL11052958 0.83
SCHEMBL11055874 0.83
SCHEMBL11058990 0.82
SCHEMBL10613005 0.80 ESR1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed