SCHEMBL11073002

SCHEMBL11073002

C=CCN(CCC)C1CCC(c2ccc(Cl)cc2)(N(CC=C)CC2CC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.36
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.33
DRD2 P14416 2/20 0.32
DRD3 P35462 2/20 0.32
HTR1A P08908 1/20 0.31
CRHR1 P34998 2/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11067219 0.90 HTR1D (0.38) KCNN4HTR1DHTR1BDRD2DRD3
SCHEMBL11070194 0.89 HTR1D (0.37) HTR1DHTR1BDRD2DRD3HTR1A
SCHEMBL11076146 0.88 HTR1D (0.36) HTR1DHTR1BDRD2DRD3HTR1A
SCHEMBL11068797 0.87 KCNN4 (0.32) KCNN4
SCHEMBL11072605 0.85 SLC6A4 (0.41) KCNN4
SCHEMBL11075429 0.84 HTR1D (0.34) HTR1DHTR1BDRD2DRD3HTR1A
SCHEMBL11075507 0.84 HTR1D (0.39) HTR1DHTR1BDRD2DRD3HTR1A
SCHEMBL11078545 0.81 KCNN4 (0.33) KCNN4CRHR1
SCHEMBL11073938 0.81 GRIN2B (0.37) KCNN4
SCHEMBL11077331 0.78 KCNN4 (0.35) KCNN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed