SCHEMBL11077358

SCHEMBL11077358

Cc1c(N(C)C)ccc([N+](=O)[O-])c1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 4/20 0.56
TDP1 Q9NUW8 3/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
KDM4E B2RXH2 2/20 0.50
GLA P06280 1/20 0.50
ALDH1A1 P00352 4/20 0.49
TSHR P16473 3/20 0.45
MAPT P10636 4/20 0.42
MAPK1 P28482 2/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTT P42858 2/20 0.42
CASP6 P55212 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
KMT2A Q03164 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2257980 0.80 TDP1 (0.64) TDP1L3MBTL1ALDH1A1TSHRMAPT
SCHEMBL3824611 0.80 TDP1 (0.64) TDP1L3MBTL1ALDH1A1TSHRMAPT
SCHEMBL29197128 0.78 TDP1 (0.57) TDP1L3MBTL1ALDH1A1TSHRMAPK1
SCHEMBL27448270 0.78 TSHR (0.62) TDP1L3MBTL1KDM4EGLAALDH1A1
SCHEMBL10654458 0.77 TDP1 (0.56) HCAR3TDP1L3MBTL1ALDH1A1TSHR
SCHEMBL1448267 0.77 TDP1 (0.56) TDP1L3MBTL1KDM4EALDH1A1TSHR
SCHEMBL31146201 0.77 TDP1 (0.56) TDP1L3MBTL1KDM4EALDH1A1TSHR
SCHEMBL11091159 0.77 TDP1 (0.56) TDP1L3MBTL1KDM4EALDH1A1TSHR
SCHEMBL3826317 0.76 TDP1 (0.62) HCAR3TDP1L3MBTL1TSHRLMNA
SCHEMBL9847247 0.75 MAPT (0.46) HCAR3TDP1KDM4EGLAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4455311-A Imidazoquinazoline derivatives which inhibit the aggregation of blood platelets, inhibit gastric secretion or have activity on the circulatory system HOFFMANN-LA ROCHE INC. (US) 1984-06-19 US disclosed
EP-0073060-A1 Imidazoquinazoline derivatives, their preparation and medicaments containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-03-02 EP disclosed