SCHEMBL11079591

SCHEMBL11079591

COc1cccc(C2(CCC#N)C=CCCC2)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.43
KDM1A O60341 1/20 0.36
SLC6A4 P31645 10/20 0.36
SLC6A2 P23975 8/20 0.36
SLC22A1 O15245 3/20 0.36
OPRM1 P35372 3/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
MEN1 O00255 1/20 0.36
SLC6A3 Q01959 1/20 0.36
ALDH1A1 P00352 1/20 0.35
FAAH O00519 1/20 0.35
NAAA Q02083 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11087953 0.88 KMT2A (0.44) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
SCHEMBL11082812 0.84 SLC6A4 (0.40) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
SCHEMBL11086716 0.84 SLC6A4 (0.40) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
SCHEMBL11090776 0.84 KDM1A (0.42) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
SCHEMBL11081659 0.82 SLC6A2 (0.44) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
SCHEMBL11081989 0.82 SLC6A4 (0.44) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
SCHEMBL11088071 0.82 KDM1A (0.40) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
SCHEMBL11115661 0.81 KDM1A (0.40) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
Hydrochloric Acid SCHEMBL11088606 0.81 UTS2R (0.44) KMT2AKDM1ASLC6A4SLC6A2SLC22A1
Hydrochloric Acid SCHEMBL11088197 0.81 SLC6A4 (0.43) KMT2AKDM1ASLC6A4SLC6A2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033156-B1 1-PHENYL-2-CYCLOHEXENE-1-ALKYLAMINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-10-17 EP disclosed
US-4448991-A ANALGESICS HOFFMANN-LA ROCHE INC. (US) 1984-05-15 US disclosed
US-4336268-A Cyclohexene derivative analgesics HOFFMANN-LA ROCHE INC. (US) 1982-06-22 US disclosed
EP-0033156-A2 1-Phenyl-2-cyclohexene-1-alkylamine derivatives, process for their preparation and medicines containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-08-05 EP disclosed