SCHEMBL11079982

SCHEMBL11079982

COCc1ccc(C23CC2C(=O)NC3=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.59
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
MMP13 P45452 1/20 0.33
CXCR3 P49682 3/20 0.33
NAAA Q02083 1/20 0.32
PTGS2 P35354 1/20 0.31
MGAT2 Q10469 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11075680 0.80 CYP19A1 (0.64) CYP19A1CXCR3
SCHEMBL12313146 0.80 CYP19A1 (0.64) CYP19A1CXCR3
SCHEMBL11911732 0.80 CYP19A1 (0.64) CYP19A1CXCR3
SCHEMBL14520901 0.79 CYP19A1 (0.72) CYP19A1CXCR3
SCHEMBL4556388 0.79 CYP19A1 (0.72) CYP19A1CXCR3
SCHEMBL8245665 0.74 CYP19A1 (0.70) CYP19A1CXCR3
SCHEMBL10530941 0.74 CYP19A1 (1.00) CYP19A1
SCHEMBL22623727 0.74 CYP19A1 (1.00) CYP19A1
SCHEMBL10530071 0.74 CYP19A1 (1.00) CYP19A1
SCHEMBL13201868 0.74 CYP19A1 (0.70) CYP19A1CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4435419-A Method of treating depression using azabicyclohexanes AMERICAN CYANAMID COMPANY (US) 1984-03-06 US disclosed
US-4231935-A ANXIOLYTICS AND ANALGESICS AMERICAN CYANAMID COMPANY (US) 1980-11-04 US disclosed
US-4196120-A 1,2-BIS(HYDROCARBYLSULFONYLOXY OR HALO METHYL)CYCLOPROPYLBENZENE, OPTICAL ACITIVITY ANALGESICS AMERICAN CYANAMID COMPANY (US) 1980-04-01 US disclosed
US-4131611-A ANXIOLYTIC, ANALGESIC AMERICAN CYANAMID COMPANY (US) 1978-12-26 US disclosed