SCHEMBL11080341

SCHEMBL11080341

Cc1ccccc1/C=C1\CCn2c1nc1ccc(N)cc1c2=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
CCR3 P51677 6/20 0.51
ALOX5 P09917 2/20 0.51
CYP1A1 P04798 1/20 0.51
CYP1B1 Q16678 1/20 0.51
HPGD P15428 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HSD17B10 Q99714 1/20 0.49
PDE4D Q08499 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080354 1.00 NPC1 (0.56) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11083270 0.92 MEN1 (0.57) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11083267 0.92 MEN1 (0.57) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11089197 0.89 MEN1 (0.58) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11089202 0.89 MEN1 (0.58) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11078402 0.88 MEN1 (0.68) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11078388 0.88 MEN1 (0.68) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11078870 0.88 CCR3 (0.64) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11078868 0.88 CCR3 (0.64) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL11081499 0.87 NPC1 (0.57) NPC1RAB9ACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4428952-A Substituted pyrrolo[2,1-b]quinazolines and pyrido[2,1-b]quinazolines useful for the treatment of or the prevention of gastrointestinal ulcers FARMITALIA CARLO ERBA S.P.A. (IT) 1984-01-31 US disclosed