SCHEMBL11100548

SCHEMBL11100548

COc1ccc(C(=O)CNCc2ccccc2)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
LMNA P02545 1/20 0.58
SMN1; SMN2 Q16637 4/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
HPGD P15428 1/20 0.56
MAPT P10636 3/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
NR1H4 Q96RI1 1/20 0.54
GAA P10253 1/20 0.54
HDAC1 Q13547 2/20 0.52
HDAC8 Q9BY41 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
BCHE P06276 1/20 0.52
ACHE P22303 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
SMPD1 P17405 1/20 0.52
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL307912 0.89 CA12 (0.56) ALDH1A1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL11437720 0.88 SMN1; SMN2 (0.70) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL11258821 0.86 SMN1; SMN2 (0.57) ALDH1A1LMNASMN1; SMN2NPC1MAPT
SCHEMBL27891607 0.85 HDAC1 (0.55) NR1H4HDAC1HDAC8HDAC6SMPD1
SCHEMBL6718805 0.81 NPC1 (0.63) ALDH1A1NPC1RAB9AMAPTMEN1
SCHEMBL1515747 0.81 NPC1 (0.63) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL28859140 0.80 NR1H4 (0.82) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL29668496 0.79 MEN1 (0.71) ALDH1A1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL28881824 0.79 MEN1 (0.71) ALDH1A1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL22551314 0.79 PTPN7 (0.46) ALDH1A1LMNASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0040956-B1 8-SUBSTITUTED 4-(3,4-DIHYDROXYPHENYL)-1,2,3,4-TETRAHYDROISOQUINOLINES SMITHKLINE BECKMAN CORPORATION (US) 1984-10-31 EP disclosed
US-4340600-A Renal dilating methods and compositions using 4-(3,4-dihydroxyphenyl)-1,2,3,4-tetrahydroisoquinolines SMITHKLINE CORPORATION (US) 1982-07-20 US disclosed
EP-0040956-A1 8-Substituted 4-(3,4-dihydroxyphenyl)-1,2,3,4-tetrahydroisoquinolines SMITHKLINE BECKMAN CORPORATION (US) 1981-12-02 EP disclosed