SCHEMBL11133307

SCHEMBL11133307

CCSc1ccc(/C=C(\C)c2ccc3c(c2)C(C)(C)CCC3(C)C)cc1.CCSc1ccc(C=O)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARG P13631 20/20 0.62
RARB P10826 18/20 0.62
RARA P10276 17/20 0.62
RXRA P19793 12/20 0.62
KDM4E B2RXH2 1/20 0.62
NPC1 O15118 1/20 0.62
CYP26A1 O43174 1/20 0.62
GMNN O75496 1/20 0.62
USP2 O75604 1/20 0.62
ALDH1A1 P00352 1/20 0.62
LMNA P02545 1/20 0.62
TP53 P04637 1/20 0.62
CYP1A2 P05177 1/20 0.62
POLB P06746 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2D6 P10635 1/20 0.62
NFKB1 P19838 1/20 0.62
CYP2C19 P33261 1/20 0.62
THPO P40225 1/20 0.62
MTOR P42345 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11133312 1.00 RARG (0.62) RARGRARBRARARXRAKDM4E
SCHEMBL11122914 0.94 RARG (0.65) RARGRARBRARARXRAKDM4E
SCHEMBL7082929 0.94 RARG (0.65) RARGRARBRARARXRAKDM4E
SCHEMBL7085635 0.88 RARG (0.78) RARGRARBRARARXRAKDM4E
SCHEMBL7085637 0.88 RARG (0.78) RARGRARBRARARXRAKDM4E
SCHEMBL8522088 0.82 RARG (0.61) RARGRARBRARARXRAKDM4E
SCHEMBL8522090 0.82 RARG (0.61) RARGRARBRARARXRAKDM4E
SCHEMBL8950121 0.81 RARG (0.60) RARGRARBRARARXRAKDM4E
SCHEMBL8950115 0.81 RARG (0.60) RARGRARBRARARXRAKDM4E
SCHEMBL11123385 0.81 RARG (0.70) RARGRARBRARARXRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0058370-B1 TETRAHYDRONAPHTHALENE AND INDAN COMPOUNDS, THEIR PRODUCTION AND PHARMACEUTICAL PREPARATIONS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-12-12 EP disclosed
EP-0058370-A1 Tetrahydronaphthalene and indan compounds, their production and pharmaceutical preparations F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-08-25 EP disclosed