SCHEMBL1114503

SCHEMBL1114503

FC(F)(F)c1cccc(Cc2noc(Cc3cccc(C(F)(F)F)c3)n2)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 8/20 0.59
KMT2A Q03164 8/20 0.59
ALDH1A1 P00352 3/20 0.58
HTT P42858 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.57
POLB P06746 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
TAAR1 Q96RJ0 1/20 0.44
S1PR1 P21453 1/20 0.44
S1PR3 Q99500 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13247786 0.84 KMT2A (0.50) MEN1KMT2AALDH1A1HTTL3MBTL1
SCHEMBL892526 0.80 KMT2A (0.47) MEN1KMT2AALDH1A1POLBSMN1; SMN2
Hydrochloric Acid SCHEMBL8435748 0.78 HTR2A (0.46) MEN1KMT2AALDH1A1HTTL3MBTL1
Hydrochloric Acid SCHEMBL8435744 0.75 HTR2A (0.45) MEN1KMT2AALDH1A1HTTL3MBTL1
SCHEMBL3237564 0.75 TAAR1 (0.64) ALDH1A1TSHRMAPK1HTR2CHTR2B
SCHEMBL4498695 0.75 GRIN1 (0.47) MEN1KMT2AALDH1A1HTTHTR2C
SCHEMBL26416251 0.74 MAPK1 (0.70) MEN1KMT2AALDH1A1HTTL3MBTL1
SCHEMBL893046 0.74 KMT2A (0.56) MEN1KMT2AALDH1A1TDP1
SCHEMBL9492711 0.74 HTR2C (0.48) HTR2CHTR2BTAAR1CYP1A2CYP3A4
SCHEMBL13731334 0.73 HTR2C (0.47) HTR2CHTR2BTAAR1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP disclosed