SCHEMBL11207320

SCHEMBL11207320

CC(C)c1c(Cc2ccc(N=C=O)cc2)cccc1N=C=O

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.51
TSHR P16473 1/20 0.51
CYP1A2 P05177 1/20 0.40
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
TRPA1 O75762 1/20 0.36
LDHA P00338 1/20 0.32
LDHB P07195 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10649255 0.81 CYP3A4 (0.56) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL27122 0.81 CYP3A4 (0.63) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL29368386 0.81 CYP3A4 (0.63) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL17912718 0.81 CYP3A4 (0.63) CYP3A4TSHRCYP1A2GABRA1GABRB2
Methyl Alcohol SCHEMBL9746439 0.80 CYP3A4 (0.58) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL2908186 0.80 CYP3A4 (0.58) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL9246394 0.79 CYP3A4 (0.67) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL17272582 0.79 CYP3A4 (0.57) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL8128748 0.78 CYP3A4 (0.56) CYP3A4TSHRCYP1A2GABRA1GABRB2
SCHEMBL28264129 0.77 CYP3A4 (0.58) CYP3A4TSHRCYP1A2GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0046556-B1 DIISOCYANATES OR MIXTURES OF DIISOCYANATES OF THE DIPHENYLMETHANE CLASS, PROCESSES FOR THEIR PREPARATION, AS WELL AS THEIR USE AS SYNTHESIS COMPONENTS IN THE MANUFACTURE OF POLYURETHANES BY THE ISOCYANATE-POLYADDITION PROCESS BAYER AG (DE) 1983-03-09 EP disclosed
EP-0046556-A1 Diisocyanates or mixtures of diisocyanates of the diphenylmethane class, processes for their preparation, as well as their use as synthesis components in the manufacture of polyurethanes by the isocyanate-polyaddition process BAYER AG (DE) 1982-03-03 EP disclosed