SCHEMBL11209354

SCHEMBL11209354

CC(C)Cn1nnc(CC(=O)O)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.51
CNR2 P34972 3/20 0.50
CNR1 P21554 1/20 0.50
PKM P14618 1/20 0.43
ATM Q13315 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP1A2 P05177 2/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
HDAC6 Q9UBN7 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
RECQL P46063 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20711333 0.85 TRPV1 (0.47) TRPV1CNR2CNR1PKMATM
SCHEMBL4409005 0.76 TRPV1 (0.53) TRPV1CNR2CNR1PKMATM
SCHEMBL14417090 0.75 TRPV1 (0.44) TRPV1CNR2CNR1PKMCYP1A2
SCHEMBL19302724 0.75 TRPV1 (0.49) TRPV1CNR2CNR1PKMATM
SCHEMBL20711268 0.73 TRPV1 (0.50) TRPV1CNR2CNR1TOP2A
SCHEMBL20711262 0.72 TRPV1 (0.47) TRPV1CNR2CNR1PKMATM
SCHEMBL7514634 0.72 KMT2A (0.43) PKMATMHSD17B10MEN1KMT2A
SCHEMBL3453024 0.72 POLB (0.39) PKMATMHSD17B10CYP1A2TP53
SCHEMBL14417089 0.71 TRPV1 (0.41) TRPV1CNR2CNR1CYP1A2USP2
SCHEMBL4403741 0.70 TRPV1 (0.48) TRPV1CNR2CNR1PKMATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0010735-B1 MAYTANSINOIDS, THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Takeda Chemical Industries, Ltd. (JP) 1983-03-23 EP disclosed
US-4248870-A MICROBIOCIDES, ANTITUMOR AGENTS, AND ANTIMITOTICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1981-02-03 US disclosed
EP-0010735-A1 Maytansinoids, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1980-05-14 EP disclosed