SCHEMBL11211989

SCHEMBL11211989

C#CCC12CCC(=O)C=C1c1c(cc(OC(C(=O)O)C(C)(C)C(=O)O)c(Cl)c1Cl)C2

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 5/20 0.34
ESR1 P03372 3/20 0.33
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11114746 0.89 ESR2 (0.44) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL11214339 0.88 ESR2 (0.46) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL11211308 0.87 ESR2 (0.34) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL11214119 0.86 ESR2 (0.36) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL11215443 0.86 ESR2 (0.48) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL11214393 0.85 ESR2 (0.49) ESR2ESR1
SCHEMBL10658184 0.85 ESR2 (0.36) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL11213888 0.84 ESR2 (0.34) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL10627600 0.84 ESR2 (0.40) ESR2ESR1CYP3A4CYP2C9TSHR
SCHEMBL11213037 0.82 ESR1 (0.42) ESR2ESR1CYP3A4CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337354-A BRAIN AND SPINAL CHORD DAMAGE MERCK & CO., INC. (US) 1982-06-29 US claimed
US-4337354-A BRAIN AND SPINAL CHORD DAMAGE MERCK & CO., INC. (US) 1982-06-29 US disclosed
US-4317922-A [(5,6,9a-Substituted-3-oxo-1,2,9,9a-tetrahydro-3H-fluoren-7-yl)oxy]alkanoic and cycloalkanoic acids and their analogs, esters, salts and derivatives MERCK & CO., INC. (US) 1982-03-02 US disclosed
US-4316043-A ANTIEDEMIC AGENTS MERCK & CO., INC. (US) 1982-02-16 US disclosed