SCHEMBL11215570

SCHEMBL11215570

BrC1Cc2ccccc2OC1c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.44
GABRA1 P14867 2/20 0.43
GABRB2 P47870 2/20 0.43
MAOB P27338 6/20 0.42
KDM4E B2RXH2 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
AR P10275 1/20 0.42
CYP19A1 P11511 1/20 0.42
HSD17B10 Q99714 1/20 0.42
AOC2 O75106 5/20 0.36
MAOA P21397 5/20 0.36
CHRM2 P08172 2/20 0.36
CHRM4 P08173 2/20 0.36
CHRM5 P08912 2/20 0.36
CHRM1 P11229 2/20 0.36
CHRM3 P20309 2/20 0.36
DAO P14920 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
DYRK1A Q13627 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16376659 0.79 CYP2C19 (0.47) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL10698516 0.79 MAOB (0.39) GABRA1GABRB2MAOBKDM4EADORA3
SCHEMBL18746282 0.78 CYP3A4 (0.48) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL1659938 0.78 CYP3A4 (0.48) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL11044980 0.78 HSP90AB1 (0.44) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL23867147 0.78 HSP90AB1 (0.44) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL460038 0.78 CYP3A4 (0.48) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL11044986 0.78 HSP90AB1 (0.44) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL1659934 0.78 CYP3A4 (0.48) HSP90AB1GABRA1GABRB2MAOBKDM4E
SCHEMBL11044983 0.78 HSP90AB1 (0.44) HSP90AB1GABRA1GABRB2MAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334067-A ANTICONVULASANTS, ANTIULCER AGENTS MARUKO SEIYAKU CO., LTD. (JP) 1982-06-08 US disclosed