SCHEMBL11218044

SCHEMBL11218044

CC(=O)Oc1cc2c(c(Cl)c1Cl)C1=CC(=O)CCC1(CC(C)C)C2

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 7/20 0.38
ESR1 P03372 5/20 0.37
TSHR P16473 2/20 0.32
HSD17B10 Q99714 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
HIF1A Q16665 1/20 0.32
LMNA P02545 1/20 0.32
BLM P54132 1/20 0.32
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
RECQL P46063 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11218826 0.90 ESR2 (0.37) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL11116181 0.88 ESR2 (0.39) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL7787631 0.87 ESR2 (0.52) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL7787618 0.87 ESR2 (0.52) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL11111591 0.86 HSD17B10 (0.48) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL10738969 0.86 ESR2 (0.51) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL11109208 0.85 ESR2 (0.53) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL11118819 0.85 ESR2 (0.38) ESR2ESR1TSHRHSD17B10MEN1
SCHEMBL11356869 0.83 ESR2 (0.54) ESR2ESR1
SCHEMBL11116986 0.83 ESR2 (0.45) ESR2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4356314-A [5,6,9A-Substituted-3-oxo-1,2,9,9a-tetrahydro-3H-fluoren-7-yl)oxy]alkanoic and cycloalkanoic acids, their analogs, esters, salts, and derivatives MERCK & CO., INC. (US) 1982-10-26 US disclosed
US-4356313-A [(5,6,9a-substituted-3-oxo-1,2,9,9a-tetrahydro-3H-fluoren-7-yl)oxy]alkanoic and cycloalkanoic acid esters and their analogs, the parent acids and their salts MERCK & CO., INC. (US) 1982-10-26 US disclosed
US-4337354-A BRAIN AND SPINAL CHORD DAMAGE MERCK & CO., INC. (US) 1982-06-29 US disclosed
US-4317922-A [(5,6,9a-Substituted-3-oxo-1,2,9,9a-tetrahydro-3H-fluoren-7-yl)oxy]alkanoic and cycloalkanoic acids and their analogs, esters, salts and derivatives MERCK & CO., INC. (US) 1982-03-02 US disclosed
US-4316043-A ANTIEDEMIC AGENTS MERCK & CO., INC. (US) 1982-02-16 US disclosed