SCHEMBL11222951

SCHEMBL11222951

Nc1cccc(Cl)c1C#CC1CCCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.45
GRM5 P41594 3/20 0.41
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.35
ALDH1A1 P00352 2/20 0.35
NR4A2 P43354 1/20 0.35
PIK3CB P42338 1/20 0.35
KDM4E B2RXH2 2/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
CREBBP Q92793 2/20 0.33
FFAR1 O14842 2/20 0.33
FFAR4 Q5NUL3 2/20 0.33
BRD4 O60885 1/20 0.33
NPSR1 Q6W5P4 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
GLA P06280 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11244447 1.00 KCNH2 (0.45) KCNH2GRM5CYP1A2TSHRALDH1A1
SCHEMBL23705829 0.92 TSHR (0.39) KCNH2GRM5CYP1A2TSHRALDH1A1
SCHEMBL30042933 0.92 TSHR (0.39) KCNH2GRM5CYP1A2TSHRALDH1A1
SCHEMBL11237060 0.88 KCNH2 (0.51) KCNH2GRM5CYP1A2TSHRALDH1A1
SCHEMBL11226503 0.88 KCNH2 (0.51) KCNH2GRM5CYP1A2TSHRALDH1A1
SCHEMBL11230085 0.86 KCNH2 (0.49) KCNH2GRM5CYP1A2ALDH1A1PIK3CB
SCHEMBL11232821 0.81 KCNH2 (0.45) KCNH2GRM5CYP1A2ALDH1A1PIK3CB
SCHEMBL11235633 0.81 KCNH2 (0.45) KCNH2GRM5CYP1A2KDM4ECREBBP
SCHEMBL11235810 0.77 KCNH2 (0.42) KCNH2GRM5CYP1A2GAACREBBP
SCHEMBL26686064 0.75 GRM5 (0.45) KCNH2GRM5CYP1A2PIK3CBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365093-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1982-12-21 US claimed
US-4096279-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain fever and inflammation WILLIAM H. RORER, INC. (US) 1978-06-20 US claimed