SCHEMBL11248052

SCHEMBL11248052

Cc1[nH]c(=O)c(N)cc1-c1ccccn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.60
PDE3A Q14432 2/20 0.60
PDE4A P27815 1/20 0.60
PDE4B Q07343 1/20 0.60
PDE4C Q08493 1/20 0.60
PDE4D Q08499 1/20 0.60
AURKB Q96GD4 2/20 0.57
INCENP Q9NQS7 2/20 0.57
CHEK1 O14757 1/20 0.47
KDM4E B2RXH2 5/20 0.41
LMNA P02545 4/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
MET P08581 1/20 0.41
BTK Q06187 2/20 0.41
HTT P42858 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11242781 0.82 CHEK1 (0.47) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11236144 0.80 BTK (0.51) CHEK1BTKBRD4IKBKB
SCHEMBL11231370 0.79 PDE3B (0.54) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11239062 0.78 KDM4E (0.50) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL7272616 0.78 KDM4E (0.63) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL6623765 0.77 KDM4E (0.53) CHEK1KDM4ELMNANPC1RAB9A
SCHEMBL8207560 0.76 PDE3B (1.00) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11232487 0.75 JAK1 (0.46) CHEK1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL11239237 0.75 PARP1 (0.40) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11246077 0.74 CHEK1 (0.48) CHEK1KDM4ELMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed