SCHEMBL11248997

SCHEMBL11248997

COc1cccc([C@@]23CCC[C@@H]2CN(C)CC3)c1

nearest known ligand 0.79

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 13/20 0.79
SLC6A2 P23975 11/20 0.73
SLC6A3 Q01959 11/20 0.73
KMT2A Q03164 1/20 0.52
CYP2D6 P10635 6/20 0.51
OPRM1 P35372 3/20 0.51
OPRD1 P41143 3/20 0.51
OPRK1 P41145 3/20 0.51
CYP2C19 P33261 2/20 0.46
KCNH2 Q12809 2/20 0.46
CYP1A1 P04798 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249000 1.00 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11251511 1.00 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
Hydrochloric Acid SCHEMBL11256706 0.99 SLC6A4 (0.77) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11078224 0.96 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11077521 0.96 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11077517 0.96 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11553658 0.95 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11553038 0.95 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11548028 0.95 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6
SCHEMBL11533791 0.91 SLC6A4 (0.79) SLC6A4SLC6A2SLC6A3KMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337341-A 4a-Aryl-octahydro-1H-2-pyrindines ELI LILLY AND COMPANY (US) 1982-06-29 US disclosed
US-4277608-A Method of preparing 4a-arylhexahydro-1H-2-pyrindines and 4a-aryloctahydroisoquinolines ELI LILLY AND COMPANY (US) 1981-07-07 US disclosed
US-4236009-A Method of preparing 4A-arylhexahydro-1H-2-pyrindines and 4A-aryloctahydroisoquinolines ELI LILLY AND COMPANY (US) 1980-11-25 US disclosed