SCHEMBL1125301

SCHEMBL1125301

O=C(O)CCc1cccc(OCc2cccc(-c3c(Cc4ccccc4)cnc4c(F)cccc34)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 7/20 0.59
NR1H3 Q13133 7/20 0.59
PPARG P37231 1/20 0.59
PPARD Q03181 1/20 0.59
PPARA Q07869 1/20 0.59
FFAR1 O14842 13/20 0.55
FFAR4 Q5NUL3 2/20 0.55
AKR1B1 P15121 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1124816 0.89 NR1H2 (0.76) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL1125566 0.82 NR1H2 (0.84) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL1125981 0.80 NR1H2 (0.70) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL1125786 0.78 NR1H2 (0.67) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL1126467 0.77 NR1H2 (0.60) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL1125913 0.76 NR1H2 (0.75) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL1125273 0.76 NR1H2 (0.90) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL1125409 0.76 NR1H2 (0.74) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL17413684 0.76 FFAR1 (0.80) FFAR1FFAR4AKR1B1
SCHEMBL14274514 0.75 NR1H2 (0.80) NR1H2NR1H3PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2284157-A1 Quinolines useful in treating cardiovascular disease Wyeth (US) 2011-02-16 EP claimed