SCHEMBL11257993

SCHEMBL11257993

Cc1cc(-c2cccnc2)nn(C)c1=O

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.57
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
CA9 Q16790 1/20 0.57
BRD4 O60885 1/20 0.52
CYP2A6 P11509 6/20 0.51
CYP2E1 P05181 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2B6 P20813 2/20 0.50
CYP2C19 P33261 2/20 0.50
ALK Q9UM73 1/20 0.46
CYP3A4 P08684 2/20 0.45
USP8 P40818 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
PIM1 P11309 1/20 0.43
PIM3 Q86V86 1/20 0.43
PIM2 Q9P1W9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053682 0.83 CYP2A6 (0.49) CA12CA1CA2CA9CYP2A6
SCHEMBL11254410 0.82 BRD4 (0.49) CA12CA1CA2CA9BRD4
SCHEMBL2689845 0.79 CYP2A6 (0.54) CA12CA1CA2CA9CYP2A6
SCHEMBL4061767 0.79 CYP2A6 (0.50) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12279439 0.79 CYP2A6 (0.54) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL28574445 0.78 CYP2A6 (0.53) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL12744778 0.78 CYP2A6 (0.53) CA12CA1CA2CA9CYP2A6
SCHEMBL15006818 0.75 CYP2A6 (0.50) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL2691331 0.75 CYP2A6 (0.50) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL17980254 0.75 MAPT (0.55) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337253-A 4,5-Dihydro-2-methyl-6-(4-pyridinyl)-3(2H)-pyridazinone and its use as a cardiotonic STERLING DRUG INC. (US) 1982-06-29 US disclosed