SCHEMBL11261876

SCHEMBL11261876

O=C(O)Cc1c(-c2ccccc2)nn(-c2ccc(Cl)c(Cl)c2)c1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
CYP1A2 P05177 1/20 0.54
GAA P10253 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
HTT P42858 1/20 0.54
PTGDR2 Q9Y5Y4 7/20 0.53
RPA1 P27694 8/20 0.51
FABP3 P05413 1/20 0.44
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11254556 0.86 PTGDR2 (0.47) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11255212 0.86 PTGDR2 (0.54) KDM4EALDH1A1CYP1A2GAACYP2D6
Trifezolac SCHEMBL11182574 0.84 KDM4E (0.51) KDM4EALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL11249550 0.83 CA1 (0.58) PTGDR2
SCHEMBL11699362 0.82 KDM4E (0.55) KDM4EALDH1A1CYP1A2GAACYP2C9
SCHEMBL11254211 0.81 CA1 (0.53) KDM4EALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL11250252 0.81 CNR1 (0.51) PTGDR2
SCHEMBL11246732 0.81 PTGDR2 (0.52) KDM4EALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL11257118 0.81 PTGDR2 (0.54) KDM4EALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL11243360 0.81 KDM4E (0.56) KDM4EALDH1A1CYP1A2GAACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4325962-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIDYRETICS BYK-GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1982-04-20 US disclosed
US-4146721-A ANALGESICS, ANTIINFLAMMATORY AGENTS AND ANTIPYRETICS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1979-03-27 US disclosed