SCHEMBL1126196

SCHEMBL1126196

COc1cc(OC)c(Cl)c(-c2ccc(C(=O)O)c3nccnc23)c1Cl.O=S(=O)(Cl)Cl

nearest known ligand 0.58

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 20/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126061 0.96 FGFR3 (0.61) FGFR3
SCHEMBL14212753 0.89 FGFR3 (0.54) FGFR3
Terephthalamide SCHEMBL3317406 0.89 FGFR3 (0.69) FGFR3
SCHEMBL1126290 0.88 FGFR3 (0.59) FGFR3
4-Aminophenol SCHEMBL3316909 0.87 FGFR3 (0.54) FGFR3
SCHEMBL1126081 0.86 FGFR3 (0.56) FGFR3
SCHEMBL3317414 0.85 FGFR3 (0.65) FGFR3
SCHEMBL3313774 0.85 FGFR3 (0.53) FGFR3
SCHEMBL4327938 0.84 FGFR3 (0.54) FGFR3
SCHEMBL3313344 0.84 FGFR3 (0.55) FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282995-A1 DERIVATIVES OF QUINOLINES AND QUINOXALINES AS PROTEIN TYROSINE KINASE INHIBITORS Novartis AG (CH) 2011-02-16 EP disclosed
WO-2009141386-A1 DERIVATIVES OF QUINOLINES AND QUINOXALINES AS PROTEIN TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2009-11-26 WO disclosed