SCHEMBL11268428

SCHEMBL11268428

CC(=O)c1cc2ccccc2cc1C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.59
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 3/20 0.58
HPGD P15428 2/20 0.58
MYC P01106 1/20 0.53
MAPT P10636 2/20 0.52
GFER P55789 1/20 0.52
NGLY1 Q96IV0 1/20 0.52
CA12 O43570 3/20 0.50
CA9 Q16790 3/20 0.50
MAOB P27338 2/20 0.50
CYP1A2 P05177 1/20 0.50
NT5E P21589 1/20 0.50
PTPN1 P18031 1/20 0.50
WDR5 P61964 1/20 0.48
ALOX15 P16050 1/20 0.48
CA1 P00915 2/20 0.47
CA4 P22748 2/20 0.47
CA5A P35218 2/20 0.47
CA7 P43166 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28466533 0.91 KDM4E (0.57) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL29373760 0.89 IDO1 (0.71) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL69178 0.89 IDO1 (0.71) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL1667141 0.86 KDM4E (0.53) IDO1ALDH1A1KDM4EHPGDMYC
Hydrochloric Acid SCHEMBL1958555 0.86 IDO1 (0.68) IDO1ALDH1A1KDM4EHPGDMYC
Hydrochloric Acid SCHEMBL28770512 0.86 IDO1 (0.68) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL12983974 0.86 IDO1 (0.68) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL29450086 0.84 IDO1 (0.65) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL69728 0.84 IDO1 (0.65) IDO1ALDH1A1KDM4EHPGDMYC
SCHEMBL9723720 0.82 IDO1 (0.63) IDO1ALDH1A1KDM4EHPGDMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020163673-A1 INHIBITORS OF ADENYLATE-FORMING ENZYME MENE MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2020-08-13 WO disclosed
US-9052654-B2 Polyamic acid composition, polyimide endless belt, and image forming apparatus FUJI XEROX CO., LTD. (JP) 2015-06-09 US disclosed
US-9052654-B2 Polyamic acid composition, polyimide endless belt, and image forming apparatus FUJI XEROX CO., LTD. (JP) 2015-06-09 US disclosed
US-8354493-B2 Polyamic acid composition, polyimide endless belt, belt supporting member, fixing member and image formation device FUJI XEROX CO., LTD. (JP) 2013-01-15 US disclosed
US-8354493-B2 Polyamic acid composition, polyimide endless belt, belt supporting member, fixing member and image formation device FUJI XEROX CO., LTD. (JP) 2013-01-15 US disclosed
US-20100233488-A1 POLYAMIC ACID COMPOSITION, POLYIMIDE ENDLESS BELT, BELT SUPPORTING MEMBER, FIXING MEMBER AND IMAGE FORMATION DEVICE FUJI XEROX CO., LTD. (JP) 2010-09-16 US disclosed
US-20100233488-A1 POLYAMIC ACID COMPOSITION, POLYIMIDE ENDLESS BELT, BELT SUPPORTING MEMBER, FIXING MEMBER AND IMAGE FORMATION DEVICE FUJI XEROX CO., LTD. (JP) 2010-09-16 US disclosed
US-20100078596-A1 POLYAMIC ACID COMPOSITION, POLYIMIDE ENDLESS BELT, AND IMAGE FORMING APPARATUS FUJI XEROX CO., LTD. (JP) 2010-04-01 US disclosed
US-20100078596-A1 POLYAMIC ACID COMPOSITION, POLYIMIDE ENDLESS BELT, AND IMAGE FORMING APPARATUS FUJI XEROX CO., LTD. (JP) 2010-04-01 US disclosed
US-4351842-A N-Cyclopropylisoindolines GLAXO LABORATORIES LIMITED (GB) 1982-09-28 US disclosed