⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL10622467 | 1.00 | — | — | |
| SCHEMBL10482149 | 1.00 | — | — | |
| SCHEMBL29761 | 0.96 | — | — | |
| SCHEMBL11127109 | 0.96 | TSHR (0.50) | — | |
| SCHEMBL672984 | 0.96 | — | — | |
| Hydrochloric Acid SCHEMBL135075 | 0.92 | — | — | |
| Iodide SCHEMBL2584329 | 0.92 | — | — | |
| Hydrogen Sulfide SCHEMBL6874931 | 0.92 | TSHR (0.46) | — | |
| SCHEMBL6372546 | 0.92 | — | — | |
| Bromide SCHEMBL5897386 | 0.92 | — | — |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 181 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-4323362-A1 | METHODS OF PREPARING CARBANUCLEOSIDES USING AMIDES | GILEAD SCIENCES, INC. (US) | 2024-02-21 | — | — | EP | claimed |
| CN-112679512-A | Tributine intermediate and preparation method thereof | 南通诺泰生物医药技术有限公司 | 2021-04-20 | — | — | CN | claimed |
| EP-3081560-B1 | TAXANES COMPOUNDS, PREPARATION METHOD THEREFOR, AND USES THEREOF | JIANGSU TASLY DIYI PHARMACEUTICAL CO LTD (CN) | 2021-03-24 | — | — | EP | claimed |
| CN-110240590-A | A kind of pyrimidine quinoline and its preparation method and application | 广州新民培林医药科技有限公司 | 2019-09-17 | — | — | CN | claimed |
| US-10253007-B2 | Taxanes compounds, preparation method therefor, and uses thereof | JIANGSU TASLY DIYI PHARMACEUTICAL CO., LTD. (CN) | 2019-04-09 | — | — | US | claimed |
| WO-2019067139-A1 | SELECTIVE REDUCTION OF CHLORODISILANES WITH TRI-N-BUTYL TIN HYDRIDE | DOW SILICONES CORPORATION (US) | 2019-04-04 | — | — | WO | claimed |
| CN-107089949-A | A kind of organotin PVC stabilizer and preparation method thereof | 毛龙飞 | 2017-08-25 | — | — | CN | claimed |
| CN-107033092-A | The preparation method of the new organo-tin compound acted on PVC stabilizer | 毛龙飞 | 2017-08-11 | — | — | CN | claimed |
| CN-107011276-A | A kind of preparation method of new organotin PVC stabilizer | 毛龙飞 | 2017-08-04 | — | — | CN | claimed |
| CN-106986836-A | The preparation method of novel techykinin antagonist with antibacterial activity | 毛阿龙 | 2017-07-28 | — | — | CN | claimed |
| CN-106966982-A | 3,5 trifluoromethylbenzenes link 1H pyrazole compounds with antibacterial activity and its preparation method and application | 毛龙飞 | 2017-07-21 | — | — | CN | claimed |
| CN-106478714-A | A kind of Alkyzin compound or the preparation method of benzyl tin compound | 北京大学 | 2017-03-08 | — | — | CN | claimed |
| EP-3081560-A1 | TAXANES COMPOUNDS, PREPARATION METHOD THEREFOR, AND USES THEREOF | Jiangsu Tasly Diyi Pharmaceutical Co., Ltd. (CN) | 2016-10-19 | — | — | EP | claimed |
| US-20160297784-A1 | Taxanes Compounds, Preparation Method Therefor, and Uses Thereof | JIANGSU TASLY DIYI PHARMACEUTICAL CO., LTD. (CN) | 2016-10-13 | — | — | US | claimed |
| CN-104650012-A | Taxane compound | TASLY HOLDING GROUP CO LTD | 2015-05-27 | — | — | CN | claimed |
| CN-101973917-B | Method for catalyzing asymmetric Michael addition through alpha, beta-unsaturated ketone and sulfonyl compound and application thereof | UNIV EAST CHINA SCIENCE & TECH | 2015-03-04 | — | — | CN | claimed |
| WO-2006007917-A1 | COMPOSITION OF FLUORINATED SILICONES, PARTICULARLY BUT NOT EXCLUSIVELY FOR ADHESIVE-RELEASING COATINGS, AND PREPARATION THEREOF | MAFLON S.R.L. (IT) | 2006-01-26 | — | — | WO | claimed |
| WO-2002072547-A1 | AMINATION PROCESS | ADVANCED RESEARCH AND TECHNOLOGY INSTITUTE, INC. (US) | 2002-09-19 | — | — | WO | claimed |
| WO-2002070439-A2 | AMINATION PROCESS | JOHNSTON, JEFFREY, N. | 2002-09-12 | — | — | WO | claimed |
| JP-6211890-A | — | — | None | — | — | JP | disclosed |
| CN-115925675-B | PSAMMAPLIN A derivatives, and preparation method and application thereof | 中国海洋大学 | 2025-04-01 | — | — | CN | disclosed |
| CN-111132985-B | Integrated process for the manufacture of methylchlorohydrosilane | 莫门蒂夫性能材料股份有限公司 | 2024-01-02 | — | — | CN | disclosed |
| US-20230414771-A1 | PREPARATION AND USE OF IMMUNOSTIMULATORY CONJUGATED COMPLEXES FOR TARGETED DELIVERY AND ACTIVATION | YAFEI SHANGHAI BIOLOGY MEDICINE SCIENCE & TECHNOLOGY CO., LTD. (CN) | 2023-12-28 | — | — | US | disclosed |
| EP-4165024-A1 | CYCLOBUTYL DIHYDROQUINOLINE SULFONAMIDE COMPOUNDS | Amgen Inc. (US) | 2023-04-19 | — | — | EP | disclosed |
| CN-115925675-A | Psamaplin A derivative and preparation method and application thereof | 中国海洋大学 | 2023-04-07 | — | — | CN | disclosed |
| CN-110997683-B | Synthesis of 1, 1-trichlorosilane | 南大光电半导体材料有限公司 | 2023-03-31 | — | — | CN | disclosed |
| EP-4108675-A1 | PREPARATION AND USE OF IMMUNOSTIMULATORY COUPLING COMPLEX WHICH IS DELIVERED AND ACTIVATED IN TARGETED MANNER | Yafei Shanghai Biolog Medicine Science & Technology Co., Ltd. (CN) | 2022-12-28 | — | — | EP | disclosed |
| WO-2021252820-A1 | CYCLOBUTYL DIHYDROQUINOLINE SULFONAMIDE COMPOUNDS | AMGEN INC. (US) | 2021-12-16 | — | — | WO | disclosed |
| CN-111647000-B | Pyrazine derivative and application thereof in inhibition of SHP2 | 勤浩医药（苏州）有限公司 | 2021-10-12 | — | — | CN | disclosed |
| CN-113474338-A | Pyrazine derivative and application thereof in inhibition of SHP2 | 勤浩医药（苏州）有限公司 | 2021-10-01 | — | — | CN | disclosed |
| WO-2021108198-A1 | INHIBITORS OF RECEPTOR INTERACTING PROTEIN KINASE I FOR THE TREATMENT OF DISEASE | BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) | 2021-06-03 | — | — | WO | disclosed |
| EP-3081560-B1 | TAXANES COMPOUNDS, PREPARATION METHOD THEREFOR, AND USES THEREOF | JIANGSU TASLY DIYI PHARMACEUTICAL CO LTD (CN) | 2021-03-24 | — | — | EP | disclosed |
| EP-3072896-B1 | TAXANE COMPOUND, AND PREPARATION METHOD AND USE THEREOF | JIANGSU TASLY DIYI PHARMACEUTICAL CO LTD (CN) | 2021-01-06 | — | — | EP | disclosed |
| CN-111647000-A | Pyrazine derivative and application thereof in inhibition of SHP2 | 勤浩医药（苏州）有限公司 | 2020-09-11 | — | — | CN | disclosed |
| CN-107417595-B | Series monoterpene indole alkaloid skeleton based on free radical tandem reaction and synthetic method of natural product | 四川大学 | 2020-07-24 | — | — | CN | disclosed |
| CN-110997683-A | Synthesis of 1,1, 1-trichlorosilane | 美国陶氏有机硅公司 | 2020-04-10 | — | — | CN | disclosed |
| CN-110240590-A | A kind of pyrimidine quinoline and its preparation method and application | 广州新民培林医药科技有限公司 | 2019-09-17 | — | — | CN | disclosed |
| US-10253007-B2 | Taxanes compounds, preparation method therefor, and uses thereof | JIANGSU TASLY DIYI PHARMACEUTICAL CO., LTD. (CN) | 2019-04-09 | — | — | US | disclosed |
| WO-2019067139-A1 | SELECTIVE REDUCTION OF CHLORODISILANES WITH TRI-N-BUTYL TIN HYDRIDE | DOW SILICONES CORPORATION (US) | 2019-04-04 | — | — | WO | disclosed |
| CN-106478714-B | A kind of preparation method of Alkyzin compound or benzyl tin compound | 北京大学 | 2019-01-18 | — | — | CN | disclosed |
| CN-104650109-B | Bearing taxanes | 江苏天士力帝益药业有限公司 | 2019-01-01 | — | — | CN | disclosed |
| CN-108558806-A | A kind of key intermediate and preparation method thereof of 5- oXo-tetrahydros pyrans -3- carboxylates | 南京药石科技股份有限公司 | 2018-09-21 | — | — | CN | disclosed |
| CN-104926712-B | Synthesize intermediate of VX-960 and preparation method thereof | 上海医药工业研究院 | 2018-03-23 | — | — | CN | disclosed |
| US-9890175-B2 | Taxane compound, and preparation method and use thereof | JIANGSU TASLY DIYI PHARMACEUTICAL CO., LTD. (CN) | 2018-02-13 | — | — | US | disclosed |
| CN-107417595-A | A kind of synthetic method of serial monoterpenoid indole alkaloid skeleton and natural products based on free radical cascade reaction | 四川大学 | 2017-12-01 | — | — | CN | disclosed |
| CN-107260733-A | The preparation method of new medicament for resisting platelet aggregation of the one kind containing 1,6 dihydropyridine 3 (2H) ketone structures | 侯茜茜 | 2017-10-20 | — | — | CN | disclosed |
| CN-107089949-A | A kind of organotin PVC stabilizer and preparation method thereof | 毛龙飞 | 2017-08-25 | — | — | CN | disclosed |
| CN-107033092-A | The preparation method of the new organo-tin compound acted on PVC stabilizer | 毛龙飞 | 2017-08-11 | — | — | CN | disclosed |
| CN-107011276-A | A kind of preparation method of new organotin PVC stabilizer | 毛龙飞 | 2017-08-04 | — | — | CN | disclosed |
| CN-106986836-A | The preparation method of novel techykinin antagonist with antibacterial activity | 毛阿龙 | 2017-07-28 | — | — | CN | disclosed |
| CN-106966982-A | 3,5 trifluoromethylbenzenes link 1H pyrazole compounds with antibacterial activity and its preparation method and application | 毛龙飞 | 2017-07-21 | — | — | CN | disclosed |
| CN-106478714-A | A kind of Alkyzin compound or the preparation method of benzyl tin compound | 北京大学 | 2017-03-08 | — | — | CN | disclosed |
| CN-106478714-A | A kind of Alkyzin compound or the preparation method of benzyl tin compound | 北京大学 | 2017-03-08 | — | — | CN | disclosed |
| CN-106257976-A | Human plasma kallikrein inhibitors | 拜奥克里斯特制药公司 | 2016-12-28 | — | — | CN | disclosed |
| US-20160340365-A1 | TAXANE COMPOUND, AND PREPARATION METHOD AND USE THEREOF | JIANGSU TASLY DIYI PHARMACEUTICAL CO., LTD. (CN) | 2016-11-24 | — | — | US | disclosed |
| EP-3087077-A1 | INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL | Merck Sharp & Dohme Corp. (US) | 2016-11-02 | — | — | EP | disclosed |
| EP-3081560-A1 | TAXANES COMPOUNDS, PREPARATION METHOD THEREFOR, AND USES THEREOF | Jiangsu Tasly Diyi Pharmaceutical Co., Ltd. (CN) | 2016-10-19 | — | — | EP | disclosed |
| US-20160297784-A1 | Taxanes Compounds, Preparation Method Therefor, and Uses Thereof | JIANGSU TASLY DIYI PHARMACEUTICAL CO., LTD. (CN) | 2016-10-13 | — | — | US | disclosed |
| EP-3072896-A1 | TAXANE COMPOUND, AND PREPARATION METHOD AND USE THEREOF | Jiangsu Tasly Diyi Pharmaceutical Co., Ltd. (CN) | 2016-09-28 | — | — | EP | disclosed |
| CN-103354808-B | Antiviral compound | ABBVIE 公司 | 2016-08-10 | — | — | CN | disclosed |
| CN-105814062-A | Spiro-oxazolones | 豪夫迈·罗氏有限公司 | 2016-07-27 | — | — | CN | disclosed |
| CN-105793266-A | Spiro-oxazolones | 豪夫迈·罗氏有限公司 | 2016-07-20 | — | — | CN | disclosed |
| CN-105693788-A | Preparation method of acetyl protection 2,6-dideoxy alpha-glucose glycol glycosides | 华东师范大学 | 2016-06-22 | — | — | CN | disclosed |
| CN-102791693-B | Hepatitis c virus inhibitors | BRISTOL-MYERS SQUIBB CO. (US) | 2016-04-13 | — | — | CN | disclosed |
| CN-102803227-B | Morpholinyl quinazolines | MERCK PATENT GMBH (DE) | 2016-01-20 | — | — | CN | disclosed |
| CN-105228983-A | The compound regulated for kinases and indication thereof | PLEXXIKON INC | 2016-01-06 | — | — | CN | disclosed |
| CN-105121454-A | C-19 modified triterpenoids with HIV maturation inhibitory activity | BRISTOL MYERS SQUIBB CO | 2015-12-02 | — | — | CN | disclosed |
| CN-105121418-A | Benzothiazol- 6 -yl acetic acid derivatives and their use for treating an hiv infection | GILEAD SCIENCES INC | 2015-12-02 | — | — | CN | disclosed |
| CN-105001165-A | Substituted diaminocarboxamide and diaminocarbonitrile pyrimidines, compositions thereof, and methods of treatment therewith | SIGNAL PHARM LLC | 2015-10-28 | — | — | CN | disclosed |
| CN-104926831-A | Telaprevir synthesis intermediate and preparation method thereof | SHANGHAI INST PHARM INDUSTRY | 2015-09-23 | — | — | CN | disclosed |
| CN-104926712-A | Telaprevir synthesis intermediate and preparation method thereof | SHANGHAI INST PHARM INDUSTRY | 2015-09-23 | — | — | CN | disclosed |
| CN-104903322-A | Antibacterial oxadiazolone derivatives | ACTELION PHARMACEUTICALS LTD | 2015-09-09 | — | — | CN | disclosed |
| WO-2015096035-A1 | INHIBITORS OF RENAL OUTER MEDULLARY POTASSIUM CHANNEL | MERCK SHARP & DOHME CORP. (US) | 2015-07-02 | — | — | WO | disclosed |
| WO-2015100147-A1 | INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL | MERCK SHARP & DOHME CORP. (US) | 2015-07-02 | — | — | WO | disclosed |
| CN-104650109-A | Taxane compound | TASLY HOLDING GROUP CO LTD | 2015-05-27 | — | — | CN | disclosed |
| CN-104650012-A | Taxane compound | TASLY HOLDING GROUP CO LTD | 2015-05-27 | — | — | CN | disclosed |
| CN-104540826-A | Spiro-fused piperidine derivatives useful as inhibitors of extrarenal potassium channels | MERCK SHARP & DOHME | 2015-04-22 | — | — | CN | disclosed |
| CN-101973917-B | Method for catalyzing asymmetric Michael addition through alpha, beta-unsaturated ketone and sulfonyl compound and application thereof | UNIV EAST CHINA SCIENCE & TECH | 2015-03-04 | — | — | CN | disclosed |
| CN-104292146-A | Telaprevir intermediate and preparation method thereof | SHANGHAI INST PHARM INDUSTRY | 2015-01-21 | — | — | CN | disclosed |
| EP-2079844-B1 | SYNTHESIS OF INIMERS AND HYPERBRANCHED POLYMERS | UNIV AKRON (US) | 2015-01-07 | — | — | EP | disclosed |
| EP-2699585-A1 | PROCESSES FOR THE MANUFACTURE OF MACROCYCLIC DEPSIPEPTIDES AND NEW INTERMEDIATES | Novartis AG (CH) | 2014-02-26 | — | — | EP | disclosed |
| WO-2013167585-A2 | RECYCLING OF ORGANOTIN COMPOUNDS | UNIVERSITEIT ANTWERPEN (BE) | 2013-11-14 | — | — | WO | disclosed |
| US-8524942-B2 | Synthesis of inimers and hyperbranched polymers | THE UNIVERSITY OF AKRON (US) | 2013-09-03 | — | — | US | disclosed |
| US-8338450-B2 | Compounds as dipeptidyl peptidase IV (DPP IV) inhibitors | LUPIN LIMITED (IN) | 2012-12-25 | — | — | US | disclosed |
| WO-2012143888-A1 | PROCESSES FOR THE MANUFACTURE OF MACROCYCLIC DEPSIPEPTIDES AND NEW INTERMEDIATES | NOVARTIS AG (CH) | 2012-10-26 | — | — | WO | disclosed |
| CN-102712646-A | RAF inhibitor compounds and methods of use thereof | ARRAY BIOPHARMA INC | 2012-10-03 | — | — | CN | disclosed |
| WO-2012033298-A3 | METHOD FOR MANUFACTURING A NOX GAS SENSOR, AND NOX GAS SENSOR MANUFACTURED USING SAME | 일진머티리얼즈 주식회사 (KR) | 2012-05-10 | — | — | WO | disclosed |
| EP-2006289-B1 | PYRAZOLE-TYPE CYANINE DYE | WAKO PURE CHEM IND LTD (JP) | 2011-11-30 | — | — | EP | disclosed |
| US-20110144321-A1 | SYNTHETIC INTERMEDIATES AND PROCESSES | BIOCRYST PHARMACEUTICALS, INC. (US) | 2011-06-16 | — | — | US | disclosed |
| EP-2313416-A2 | SYNTHETIC INTERMEDIATES AND PROCESSES | BIOCRYST PHARMACEUTICALS, INC. (US) | 2011-04-27 | — | — | EP | disclosed |
| US-20110053856-A1 | METABOLITE DERIVATIVES OF THE HDAC INHIBITOR FK228 | GLOUCESTER PHARMACEUTICALS, INC. | 2011-03-03 | — | — | US | disclosed |
| US-20110046334-A1 | SYNTHESIS OF INIMERS AND HYPERBRANCHED POLYMERS | THE UNIVERSITY OF AKRON (US) | 2011-02-24 | — | — | US | disclosed |
| EP-2282636-A2 | BENZENE SULFONAMIDE THIAZOLE AND OXAZOLE COMPOUNDS | GlaxoSmithKline LLC (US) | 2011-02-16 | — | — | EP | disclosed |
| US-20100291020-A1 | NOVEL COMPOUNDS AS DIPEPTIDYL PEPTIDASE IV (DPP IV) INHIBITORS | LUPIN LIMITED (IN) | 2010-11-18 | — | — | US | disclosed |
| US-7709469-B2 | P2X7 receptor antagonists and methods of use | ABBOTT LABORATORIES (US) | 2010-05-04 | — | — | US | disclosed |
| US-7709636-B2 | Pyrazole sulfonylurea compound and herbicide | NISSAN CHEMICAL INDUSTRIES, LTD. (JP) | 2010-05-04 | — | — | US | disclosed |
| WO-2010011748-A2 | SYNTHETIC INTERMEDIATES AND PROCESSES | BIOCRYST PHARMACEUTICALS, INC. (US) | 2010-01-28 | — | — | WO | disclosed |
| US-20100016584-A1 | Pyrazole sulfonylurea compound and herbicide | NISSAN CHEMICAL INDUSTRIES, LTD. (JP) | 2010-01-21 | — | — | US | disclosed |
| WO-2009137391-A2 | BENZENE SULFONAMIDE THIAZOLE AND OXAZOLE COMPOUNDS | SMITHKLINE BEECHAM CORPORATION (US) | 2009-11-12 | — | — | WO | disclosed |
| EP-2079844-A1 | SYNTHESIS OF INIMERS AND HYPERBRANCHED POLYMERS | The University of Akron (US) | 2009-07-22 | — | — | EP | disclosed |
| US-7557067-B2 | Pyrazole sulfonylurea compound and herbicide | NISSAN CHEMICAL INDUSTRIES, LTD. (JP) | 2009-07-07 | — | — | US | disclosed |
| WO-2009037719-A1 | NOVEL COMPOUNDS AS DIPEPTIDYL PEPTIDASE IV (DPP IV) INHIBITORS | LUPIN LIMITED (IN) | 2009-03-26 | — | — | WO | disclosed |
| EP-2006289-A1 | PYRAZOLE-TYPE CYANINE DYE | Wako Pure Chemical Industries, Ltd. (JP) | 2008-12-24 | — | — | EP | disclosed |
| EP-1951689-A1 | P2X7 RECEPTOR ANTAGONISTS AND METHODS OF USE | ABBOTT LABORATORIES (US) | 2008-08-06 | — | — | EP | disclosed |
| EP-1924553-A1 | BICYCLO[2.2.]HEPT-7-YLAMINE DERIVATIVES AND THEIR USES | Argenta Discovery Limited (GB) | 2008-05-28 | — | — | EP | disclosed |
| WO-2008045299-A1 | SYNTHESIS OF INIMERS AND HYPERBRANCHED POLYMERS | UNIVERSITY OF AKRON (US) | 2008-04-17 | — | — | WO | disclosed |
| US-20080064600-A1 | Pyrazole Sulfonylurea Compound and Herbicide | NISSAN CHEMICAL INDUSTRIES, LTD. (JP) | 2008-03-13 | — | — | US | disclosed |
| US-20070265242-A1 | Novel Carbapenem Compound | DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) | 2007-11-15 | — | — | US | disclosed |
| US-20070129290-A1 | Metabolite derivatives of the HDAC inhibitor FK228 | GLOUCESTER PHARMACEUTICALS, INC. | 2007-06-07 | — | — | US | disclosed |
| WO-2007056046-A1 | P2X7 RECEPTOR ANTAGONISTS AND METHODS OF USE | ABBOTT LABORATORIES (US) | 2007-05-18 | — | — | WO | disclosed |
| EP-1785426-A1 | NOVEL CARBAPENEM COMPOUND | Dainippon Sumitomo Pharma Co., Ltd. (JP) | 2007-05-16 | — | — | EP | disclosed |
| US-20070105842-A1 | P2X7 receptor antagonists and methods of use | ABBVIE INC. | 2007-05-10 | — | — | US | disclosed |
| WO-2007017670-A1 | BICYCLO[2.2.]HEPT-7-YLAMINE DERIVATIVES AND THEIR USES | ARGENTA DISCOVERY LTD. (GB) | 2007-02-15 | — | — | WO | disclosed |
| EP-1748047-A1 | PYRAZOLE SULFONYLUREA COMPOUND AND HERBICIDE | Nissan Chemical Industries, Ltd. (JP) | 2007-01-31 | — | — | EP | disclosed |
| EP-1730165-A1 | INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE | SCHERING CORPORATION (US) | 2006-12-13 | — | — | EP | disclosed |
| EP-1684754-A1 | HMG-COA REDUCTASE INHIBITORS AND METHOD | Bristol-Myers Squibb Company (US) | 2006-08-02 | — | — | EP | disclosed |
| EP-1626720-A1 | 4-(2-PHENYLSULFANYL-PHENYL)-PIPERIDINE DERIVATIVES AS SEROTONIN REUPTAKE INHIBITORS | H. Lundbeck A/S (DK) | 2006-02-22 | — | — | EP | disclosed |
| WO-2006007917-A1 | COMPOSITION OF FLUORINATED SILICONES, PARTICULARLY BUT NOT EXCLUSIVELY FOR ADHESIVE-RELEASING COATINGS, AND PREPARATION THEREOF | MAFLON S.R.L. (IT) | 2006-01-26 | — | — | WO | disclosed |
| WO-2005092907-A2 | MONOSACCHARIDE DERIVATIVES AS ANTI-CANCER AND ANTI-INFLAMMATORY AGENTS | RANBAXY LABORATORIES LIMITED (IN) | 2005-10-06 | — | — | WO | disclosed |
| WO-2005085275-A1 | INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE | SCHERING CORPORATION (US) | 2005-09-15 | — | — | WO | disclosed |
| WO-2005051386-A1 | HMG-COA REDUCTASE INHIBITORS AND METHOD | BRISTOL-MYERS SQUIBB COMPANY (US) | 2005-06-09 | — | — | WO | disclosed |
| WO-2005048956-A2 | ESTRADIOL-RELATED COMPOUNDS AND METHODS OF USE AS ANTI-TUMOR AGENTS | UNIVERSITY OF MASSACHUSETTS (US) | 2005-06-02 | — | — | WO | disclosed |
| EP-1467730-A1 | NON-STEROIDAL LIGANDS FOR THE GLUCOCORTICOID RECEPTOR, COMPOSITIONS AND USES THEREOF | THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) | 2004-10-20 | — | — | EP | disclosed |
| WO-2004087156-A1 | 4-(2-PHENYLSULFANYL-PHENYL)-PIPERIDINE DERIVATIVES AS SEROTONIN REUPTAKE INHIBITORS | H. LUNDBECK A/S (DK) | 2004-10-14 | — | — | WO | disclosed |
| WO-2003061651-A1 | NON-STEROIDAL LIGANDS FOR THE GLUCOCORTICOID RECEPTOR, COMPOSITIONS AND USES THEREOF | THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) | 2003-07-31 | — | — | WO | disclosed |
| EP-1289966-A1 | SUBSTITUTED LACTAMS AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION | Bristol-Myers Squibb Pharma Company (US) | 2003-03-12 | — | — | EP | disclosed |
| WO-2002072547-A1 | AMINATION PROCESS | ADVANCED RESEARCH AND TECHNOLOGY INSTITUTE, INC. (US) | 2002-09-19 | — | — | WO | disclosed |
| WO-2002070439-A2 | AMINATION PROCESS | JOHNSTON, JEFFREY, N. | 2002-09-12 | — | — | WO | disclosed |
| EP-1232166-A2 | SYNTHESIS OF 2'-DEOXY-L-NUCLEOSIDES | Pharmasset Limited (US) | 2002-08-21 | — | — | EP | disclosed |
| EP-1204659-A2 | SEROTONERGIC BENZOFURANS | ELI LILLY AND COMPANY (US) | 2002-05-15 | — | — | EP | disclosed |
| EP-1204660-A1 | SEROTONERGIC BENZOTHIOPHENES | ELI LILLY AND COMPANY (US) | 2002-05-15 | — | — | EP | disclosed |
| EP-1202999-A1 | NOVEL 2-DECARBOXY-2-PHOSPHINICO PROSTAGLANDIN F ANALOGS | THE PROCTER & GAMBLE COMPANY (US) | 2002-05-08 | — | — | EP | disclosed |
| EP-1007031-A4 | 4-CYANO-4-DEFORMYLSORDARIN DERIVATIVES | MERCK & CO INC (US) | 2001-10-24 | — | — | EP | disclosed |
| WO-2001077086-A1 | SUBSTITUTED LACTAMS AS INHIBITORS OF Aβ PROTEIN PRODUCTION | DUPONT PHARMACEUTICALS COMPANY (US) | 2001-10-18 | — | — | WO | disclosed |
| WO-2001034618-A2 | SYNTHESIS OF 2'-DEOXY-L-NUCLEOSIDES | PHARMASSET LIMITED (US) | 2001-05-17 | — | — | WO | disclosed |
| WO-2001010873-A1 | NOVEL 2-DECARBOXY-2-PHOSPHINICO PROSTAGLANDIN F ANALOGS | THE PROCTER & GAMBLE COMPANY (US) | 2001-02-15 | — | — | WO | disclosed |
| WO-2001009126-A1 | SEROTONERGIC BENZOTHIOPHENES | ELI LILLY AND COMPANY (US) | 2001-02-08 | — | — | WO | disclosed |
| WO-2001009122-A2 | SEROTONERGIC BENZOFURANS | ELI LILLY AND COMPANY (US) | 2001-02-08 | — | — | WO | disclosed |
| EP-1007031-A1 | 4-CYANO-4-DEFORMYLSORDARIN DERIVATIVES | Merck & Co., Inc. (US) | 2000-06-14 | — | — | EP | disclosed |
| EP-1005445-A1 | N-ALKANOYLPHENYLALANINE DERIVATIVES | F. HOFFMANN-LA ROCHE AG (CH) | 2000-06-07 | — | — | EP | disclosed |
| EP-1005446-A1 | N-AROYLPHENYLALANINE DERIVATIVES | F. HOFFMANN-LA ROCHE AG (CH) | 2000-06-07 | — | — | EP | disclosed |
| EP-0915881-A1 | PYRROLOAZEPINE COMPOUNDS | SUNTORY LIMITED (JP) | 1999-05-19 | — | — | EP | disclosed |
| WO-1999010313-A1 | N-AROYLPHENYLALANINE DERIVATIVES | F.HOFFMANN-LA ROCHE AG (CH) | 1999-03-04 | — | — | WO | disclosed |
| WO-1999010312-A1 | N-ALKANOYLPHENYLALANINE DERIVATIVES | F. HOFFMANN-LA ROCHE AG (CH) | 1999-03-04 | — | — | WO | disclosed |
| WO-1999009974-A1 | 4-CYANO-4-DEFORMYLSORDARIN DERIVATIVES | MERCK & CO., INC. (US) | 1999-03-04 | — | — | WO | disclosed |
| WO-1998041527-A1 | PYRROLOAZEPINE COMPOUNDS | SUNTORY LIMITED (JP) | 1998-09-24 | — | — | WO | disclosed |
| WO-1998005662-A1 | CONFORMATIONALLY LOCKED NUCLEOSIDE ANALOGS AS ANTIHERPETIC AGENTS | THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 1998-02-12 | — | — | WO | disclosed |
| EP-0784628-A1 | INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME | Vertex Pharmaceuticals Incorporated (US) | 1997-07-23 | — | — | EP | disclosed |
| CN-1151737-A | 1, 2, 4, 6-thiatriazines with herbicidal activity | CIBA GEIGY AG (CH) | 1997-06-11 | — | — | CN | disclosed |
| EP-0737202-A1 | HYPOCHOLESTEROLEMIC AGENTS | PFIZER INC. (US) | 1996-10-16 | — | — | EP | disclosed |
| EP-0737203-A1 | STEROIDAL GLYCOSIDES | PFIZER INC. (US) | 1996-10-16 | — | — | EP | disclosed |
| US-5502073-A | INSECTICIDES OR ANTHELMINTICS | THE WELLCOME FOUNDATION (GB) | 1996-03-26 | — | — | US | disclosed |
| WO-1995035308-A1 | INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME | VERTEX PHARMACEUTICALS INCORPORATED (US) | 1995-12-28 | — | — | WO | disclosed |
| WO-1995018143-A1 | HYPOCHOLESTEROLEMIC AGENTS | PFIZER INC. (US) | 1995-07-06 | — | — | WO | disclosed |
| WO-1995018144-A1 | STEROIDAL GLYCOSIDES | PFIZER INC. (US) | 1995-07-06 | — | — | WO | disclosed |
| EP-0346427-B1 | MACROCYCLIC COMPOUNDS | FISONS PLC (GB) | 1995-03-29 | — | — | EP | disclosed |
| US-5376663-A | Immunosuppressive agents; e.g. 1,14-Dihydroxy-12-[2-(4-hydroxy-3-methoxycyclohexyl)-1-methylvinyl]-23,25-dimethoxy-13,19,21,27-tetramethyl-17-(2-oxopropyl)-11,28,-dioxa-4-azatricyclo(22.3.1.04,9)octacos-18-ene-2,3,10,16-tetraone | FISONS PLC (GB) | 1994-12-27 | — | — | US | disclosed |
| JP-H06211890-A | 2'-DEOXY-2'@(3754/24)S)-SUBSTITUTED ALKYLCYTIDINE DERIVATIVE | YAMASA SHOYU CO LTD | 1994-08-02 | — | — | JP | disclosed |
| EP-0607400-A1 | Fluorinated 17-beta substituted-4-aza-5-alpha- andostran-3one derivatives. | PHARMACIA & UPJOHN S.p.A. (IT) | 1994-07-27 | — | — | EP | disclosed |
| EP-0582338-A2 | 17-Spiromethylene steroids | Akzo Nobel N.V. (NL) | 1994-02-09 | — | — | EP | disclosed |
| US-5210227-A | IMMUNOSUPPRESSIVE COMPOUNDS | FISONS PLC (GB) | 1993-05-11 | — | — | US | disclosed |
| US-5204330-A | ANTIFUNGAL COMPOUNDS | BEECHAM GROUP P.L.C. (GB) | 1993-04-20 | — | — | US | disclosed |
| WO-1992015598-A1 | PROCESS FOR THE DEOXYGENATION OF NUCLEOSIDES | UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) | 1992-09-17 | — | — | WO | disclosed |
| EP-0439556-A4 | HETEROCYCLIC PEPTIDE RENIN INHIBITORS | — | 1991-10-30 | — | — | EP | disclosed |
| EP-0444829-A2 | Immunosuppressive compounds | FISONS plc (GB) | 1991-09-04 | — | — | EP | disclosed |
| EP-0439556-A1 | HETEROCYCLIC PEPTIDE RENIN INHIBITORS | ABBOTT LABORATORIES (US) | 1991-08-07 | — | — | EP | disclosed |
| EP-0431870-A1 | Amphotericin B derivatives | Beecham Group p.l.c. (GB) | 1991-06-12 | — | — | EP | disclosed |
| EP-0430579-A2 | Fluoroaliphatic-group-substituted esters and method of making the same | MINNESOTA MINING AND MANUFACTURING COMPANY (US) | 1991-06-05 | — | — | EP | disclosed |
| US-4937259-A | Antihypercholesterolemic compounds | MERCK & CO., INC. (US) | 1990-06-26 | — | — | US | disclosed |
| WO-1990004917-A1 | HETEROCYCLIC PEPTIDE RENIN INHIBITORS | ABBOTT LABORATORIES (US) | 1990-05-17 | — | — | WO | disclosed |
| US-4923867-A | Synthetic marcfortine derivatives useful as antiparasitic agents | MERCK & CO., INC. (US) | 1990-05-08 | — | — | US | disclosed |
| EP-0346427-A1 | MACROCYCLIC COMPOUNDS. | FISONS PLC (GB) | 1989-12-20 | — | — | EP | disclosed |
| WO-1989007102-A1 | NULCEOSIDETYPE COMPOUNDS WHICH ARE PHOSPHODIESTERASE INHIBITORS | SCHERING CORPORATION (US) | 1989-08-10 | — | — | WO | disclosed |
| EP-0324562-A1 | 1-Carba(dethia)-3-cephem derivatives | ELI LILLY AND COMPANY (US) | 1989-07-19 | — | — | EP | disclosed |
| EP-0323042-A1 | Process to macrocyclic compounds | FISONS plc (GB) | 1989-07-05 | — | — | EP | disclosed |
| WO-1989005304-A1 | MACROCYCLIC COMPOUNDS | FISONS PLC (GB) | 1989-06-15 | — | — | WO | disclosed |
| EP-0294229-A2 | Novel heterocyclic pesticidal compounds | THE WELLCOME FOUNDATION LIMITED (GB) | 1988-12-07 | — | — | EP | disclosed |
| EP-0074599-A1 | 5,6-cis-Carbapenem derivatives, their production and use | Takeda Chemical Industries, Ltd. (JP) | 1983-03-23 | — | — | EP | disclosed |
| EP-0073451-A2 | Carbapenam compound and processes for the preparation thereof | FUJISAWA PHARMACEUTICAL CO., LTD. (JP) | 1983-03-09 | — | — | EP | disclosed |
| EP-0001715-A2 | Azetidinone antibiotics and their pharmaceutical formulations and use | ELI LILLY AND COMPANY (US) | 1979-05-02 | — | — | EP | disclosed |
| US-4087447-A | Anti-secretory prostaglandins intermediates | G. D. SEARLE & CO. (US) | 1978-05-02 | — | — | US | disclosed |
| US-4087447-A | Anti-secretory prostaglandins intermediates | G. D. SEARLE & CO. (US) | 1978-05-02 | — | — | US | disclosed |