SCHEMBL11278033

SCHEMBL11278033

CCc1nn(C)c2[nH]c(=O)c3ccccc3c12

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.56
KDM4D Q6B0I6 1/20 0.43
TNKS2 Q9H2K2 1/20 0.41
CYP1A2 P05177 2/20 0.40
KDM4E B2RXH2 3/20 0.39
HSD17B10 Q99714 1/20 0.39
ALOX15 P16050 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
AURKA O14965 1/20 0.37
PDE5A O76074 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1720121 0.85 PARP1 (0.53) PARP1CYP1A2KDM4E
SCHEMBL1720598 0.83 PARP1 (0.49) PARP1KDM4EALOX15SMN1; SMN2
SCHEMBL1719750 0.81 PARP1 (0.56) PARP1KDM4E
SCHEMBL4068289 0.80 PARP1 (0.55) PARP1KDM4E
SCHEMBL1720503 0.80 PARP1 (0.55) PARP1
SCHEMBL1720862 0.80 PARP1 (0.55) PARP1
SCHEMBL1719969 0.80 PARP1 (0.53) PARP1CYP1A2KDM4EHSD17B10CYP2C9
Hydrochloric Acid SCHEMBL1719747 0.79 PARP1 (0.54) PARP1KDM4E
SCHEMBL1720304 0.79 PARP1 (0.53) PARP1KDM4EHSD17B10SMN1; SMN2
SCHEMBL1719833 0.78 PARP1 (0.49) PARP1KDM4EHSD17B10SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4113731-A PHOTOGRAPHIC EMULSION STABILIZERS GRUPPO LEPETIT S.P.A. (IT) 1978-09-12 US claimed
EP-0005745-B1 PYRAZOLO (3,4-C) AND THIAZOLO (5,4-C) ISOQUINOLINES, METHODS FOR PREPARING THEM, THESE COMPOUNDS FOR USE AS ANTIINFLAMMATORY, CNS-DEPRESSANT AND ANTI-ANXIETY AGENTS AND PHARMACEUTICAL COMPOSITIONS THEREOF GRUPPO LEPETIT S.P.A. (IT) 1982-07-14 EP disclosed
US-4232017-A CNS DEPRESSANTS; TRANQUILIZERS GRUPPO LEPETIT S.P.A. (IT) 1980-11-04 US disclosed
EP-0005745-A1 Pyrazolo (3,4-c) and thiazolo (5,4-c) isoquinolines, methods for preparing them, these compounds for use as antiinflammatory, CNS-depressant and anti-anxiety agents and pharmaceutical compositions thereof GRUPPO LEPETIT S.P.A. (IT) 1979-12-12 EP disclosed
US-4113731-A PHOTOGRAPHIC EMULSION STABILIZERS GRUPPO LEPETIT S.P.A. (IT) 1978-09-12 US disclosed