SCHEMBL11280869

SCHEMBL11280869

C/N=C(\NC)NC(=O)Nc1c(C)cccc1C

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.84
DRD2 P14416 1/20 0.67
HTR2A P28223 1/20 0.67
HTR2B P41595 1/20 0.67
PKM P14618 1/20 0.65
ATM Q13315 1/20 0.49
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
ALOX15 P16050 1/20 0.45
HTT P42858 1/20 0.45
RAB9A P51151 1/20 0.45
HSD17B10 Q99714 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
EPHX1 P07099 1/20 0.44
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11280882 1.00 POLB (0.84) POLBDRD2HTR2AHTR2BPKM
Hydrochloric Acid SCHEMBL11562609 0.98 POLB (0.82) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11558226 0.90 POLB (0.68) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11560061 0.90 POLB (0.68) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11562714 0.89 POLB (0.67) POLBDRD2HTR2AHTR2BPKM
Hydrochloric Acid SCHEMBL11560896 0.82 POLB (0.75) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11560231 0.81 CACNA1C (0.62) POLBDRD2HTR2AHTR2BPKM
SCHEMBL10937736 0.81 POLB (0.60) POLBDRD2HTR2AHTR2BPKM
SCHEMBL10937733 0.81 POLB (0.60) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11272212 0.81 POLB (0.55) POLBDRD2HTR2AHTR2BPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed