SCHEMBL1129003

SCHEMBL1129003

CC(C)(C)C(=O)N1CCC(n2ncc3c(Oc4ccc(S(C)(=O)=O)cc4)ncnc32)CC1.CC(C)(C)C(=O)N1CCC(n2ncc3c(Oc4ccc(S(C)(=O)=O)cc4)ncnc32)CC1

nearest known ligand 0.81

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.81
CYP2C9 P11712 1/20 0.54
GPR119 Q8TDV5 16/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4354573 1.00 CYP3A4 (0.81) CYP3A4CYP2C9GPR119
SCHEMBL1128529 0.92 CYP3A4 (0.77) CYP3A4CYP2C9GPR119
SCHEMBL9006352 0.90 CYP3A4 (0.79) CYP3A4CYP2C9GPR119
SCHEMBL2019784 0.90 CYP3A4 (0.79) CYP3A4CYP2C9GPR119
SCHEMBL1128644 0.90 CYP3A4 (1.00) CYP3A4CYP2C9GPR119
SCHEMBL1128844 0.89 CYP3A4 (0.84) CYP3A4CYP2C9GPR119
SCHEMBL4355890 0.89 CYP3A4 (0.77) CYP3A4CYP2C9GPR119
SCHEMBL9007710 0.88 CYP3A4 (0.64) CYP3A4CYP2C9GPR119
SCHEMBL4361119 0.88 CYP3A4 (0.75) CYP3A4CYP2C9GPR119
SCHEMBL1128902 0.88 CYP3A4 (0.75) CYP3A4CYP2C9GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283019-A1 GPR119 RECEPTOR AGONISTS F. Hoffmann-La Roche AG (CH) 2011-02-16 EP disclosed