SCHEMBL11297694

SCHEMBL11297694

N[C@@](CF)(Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 15/20 0.40
NMBR P28336 1/20 0.36
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
HIF1A Q16665 1/20 0.32
ENPP2 Q13822 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10978566 0.88 SIRT2 (0.48) SIRT2NMBR
SCHEMBL6943555 0.82 SIRT2 (0.49) SIRT2NMBRCYP11B1CYP11B2ENPP2
SCHEMBL10976975 0.80 SIRT2 (0.43) SIRT2NMBRCYP11B1CYP11B2ENPP2
SCHEMBL2002061 0.79 SIRT2 (0.45) SIRT2NMBRCYP11B1CYP11B2HIF1A
SCHEMBL31370665 0.76 SIRT2 (0.48) SIRT2NMBRENPP2
SCHEMBL877052 0.76 SIRT2 (0.46) SIRT2NMBRCYP11B1CYP11B2ENPP2
SCHEMBL10187011 0.74 SIRT2 (0.46) SIRT2NMBRCYP11B1CYP11B2ENPP2
SCHEMBL30547297 0.74 SIRT2 (0.45) SIRT2NMBRCYP11B1CYP11B2
SCHEMBL2180673 0.73 SIRT2 (0.45) SIRT2NMBRCYP11B1CYP11B2ENPP2
SCHEMBL1924923 0.73 SIRT2 (0.45) SIRT2NMBRCYP11B1CYP11B2ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0046290-A1 Synergistic combination of (R,S)alpha-fluoromethylhistidine and cimetidine as an anti-ulcer agent MERCK & CO. INC. (US) 1982-02-24 EP disclosed