SCHEMBL11314219

SCHEMBL11314219

CC(=O)c1ccc(-c2cc(F)ccc2F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.54
KIF11 P52732 1/20 0.49
MAOB P27338 4/20 0.48
HSD17B1 P14061 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
MAOA P21397 1/20 0.42
BCL2L1 Q07817 1/20 0.41
BAD Q92934 1/20 0.41
SYK P43405 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MAP4K4 O95819 1/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
ALOX5 P09917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1226198 0.89 PTGS1 (0.54) PTGS1KIF11MAOBHSD17B1SMN1; SMN2
SCHEMBL10436026 0.86 MAOB (0.55) PTGS1KIF11MAOBHSD17B1SMN1; SMN2
SCHEMBL30747689 0.86 MAOB (0.55) PTGS1KIF11MAOBHSD17B1SMN1; SMN2
SCHEMBL2555397 0.84 MAPT (0.48) PTGS1KIF11MAOBHSD17B1SMN1; SMN2
SCHEMBL22926305 0.84 FASN (0.51) PTGS1KIF11MAOBHSD17B1SMN1; SMN2
SCHEMBL16156050 0.84 PTGS1 (0.53) PTGS1KIF11MAOBHSD17B1SMN1; SMN2
SCHEMBL1222849 0.84 BCL2L1 (0.62) SMN1; SMN2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL4991368 0.82 PTGS1 (0.54) PTGS1MAPTALDH1A1MAP4K4
SCHEMBL26116358 0.81 PTGS1 (0.57) PTGS1SMN1; SMN2MAPTKDM4EMEN1
SCHEMBL2556102 0.81 PTGS1 (0.50) PTGS1KIF11MAOBHSD17B1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295402-B1 Antibacterial agents UNIV WASHINGTON (US) 2015-08-12 EP disclosed
US-4301313-A ANTIINFLAMMATORY AGENTS, ANTIPYRETICS, ANALGESICS ELI-LILLY AND COMPANY (US) 1981-11-17 US disclosed
US-4226887-A P-BIPHENYLYLACETYLENE ELI LILLY AND COMPANY (US) 1980-10-07 US disclosed
US-3991212-A PHENYLACETYLENE COMPOUNDS ELI LILLY AND COMPANY (US) 1976-11-09 US disclosed
US-3968251-A Arylacetylene compounds as antithrombotic agents ELI LILLY AND COMPANY (US) 1976-07-06 US disclosed