SCHEMBL11324364

SCHEMBL11324364

CC(C)(C)C#Cc1ccccc1Cl.CCCCCC#Cc1ccccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.45
TSHR P16473 1/20 0.45
KCNH2 Q12809 3/20 0.40
CYP2C9 P11712 4/20 0.40
CYP2C19 P33261 4/20 0.40
CYSLTR2 Q9NS75 1/20 0.39
CYSLTR1 Q9Y271 1/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
LMNA P02545 1/20 0.37
APEX1 P27695 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PGK1 P00558 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921661 0.89 KCNH2 (0.47) CYP3A4TSHRKCNH2CYP2C9CYP2C19
SCHEMBL11231181 0.88 KCNH2 (0.50) CYP3A4TSHRKCNH2CYP2C9CYP2C19
SCHEMBL11240545 0.88 KCNH2 (0.50) CYP3A4TSHRKCNH2CYP2C9CYP2C19
SCHEMBL11227888 0.85 CYP3A4 (0.47) CYP3A4TSHRKCNH2CYP2C9CYP2C19
SCHEMBL1921804 0.81 KCNH2 (0.48) TSHRKCNH2LMNAGRM5FFAR1
SCHEMBL11234645 0.78 KCNH2 (0.46) CYP3A4TSHRKCNH2CYP2C9CYP2C19
SCHEMBL6371432 0.76 KCNH2 (0.58) CYP3A4TSHRKCNH2CYP2C9CYP2C19
SCHEMBL10812341 0.72 KCNH2 (0.50) CYP3A4TSHRKCNH2CYP2C9CYP2C19
SCHEMBL6297820 0.72 KDM4E (0.57) CYP3A4KCNH2CYP2C9CYP2C19KDM4E
SCHEMBL11237484 0.70 KCNH2 (0.48) CYP3A4TSHRKCNH2CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4264627-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1981-04-28 US disclosed