SCHEMBL1133384

SCHEMBL1133384

CC(=O)OC(C)(C)c1ccccc1C(CCSCC1CC1)c1cccc(/C=C/c2ccc3ccc(Cl)cc3n2)c1.[NaH]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYSLTR1 Q9Y271 4/20 0.50
CYSLTR2 Q9NS75 3/20 0.49
CYP2C8 P10632 2/20 0.49
MEN1 O00255 1/20 0.49
RECQL P46063 1/20 0.49
BLM P54132 1/20 0.49
KMT2A Q03164 1/20 0.49
ABCB11 O95342 1/20 0.49
EGFR P00533 1/20 0.49
ESR1 P03372 1/20 0.49
NR3C1 P04150 1/20 0.49
FYN P06241 1/20 0.49
PGR P06401 1/20 0.49
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADRA2A P08913 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
CHRM1 P11229 1/20 0.49
ADRB3 P13945 1/20 0.49
ADRA2B P18089 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5708955 0.99 CYSLTR1 (0.51) CYSLTR1CYSLTR2CYP2C8MEN1RECQL
Acetic Acid SCHEMBL1133386 0.90 CYSLTR1 (0.55) CYSLTR1CYSLTR2CYP2C8MEN1RECQL
Acetic Acid SCHEMBL8610827 0.89 CYSLTR1 (0.51) CYSLTR1CYSLTR2CYP2C8MEN1RECQL
Acetic Acid SCHEMBL8594831 0.89 CYSLTR1 (0.51) CYSLTR1CYSLTR2CYP2C8MEN1RECQL
Acetic Acid SCHEMBL15475212 0.86 CYSLTR1 (0.52) CYSLTR1CYSLTR2CYP2C8MEN1RECQL
SCHEMBL23728918 0.85 CYSLTR1 (0.48) CYSLTR1CYSLTR2MEN1RECQLBLM
SCHEMBL2785946 0.85 CYSLTR1 (0.48) CYSLTR1CYSLTR2MEN1RECQLBLM
SCHEMBL20490657 0.85 CYSLTR2 (0.52) CYSLTR1CYSLTR2
SCHEMBL5521192 0.85 CYSLTR2 (0.52) CYSLTR1CYSLTR2
SCHEMBL524722 0.85 CYSLTR2 (0.52) CYSLTR1CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2287154-A1 Efficient synthesis for the preparation of montelukast KRKA, D.D., Novo Mesto (SI) 2011-02-23 EP disclosed